SCHEMBL24695415

SCHEMBL24695415

Brc1cnc(N[C@@H]2CCCNC2)nn1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 17/20 0.47
CCNK O75909 17/20 0.47
CDK9 P50750 17/20 0.47
CDK12 Q9NYV4 17/20 0.47
CCNE1 P24864 14/20 0.47
CDK2 P24941 14/20 0.47
CDK7 P50613 11/20 0.42
CCNH P51946 10/20 0.42
MNAT1 P51948 9/20 0.42
CRBN Q96SW2 1/20 0.42
CHEK1 O14757 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL268925 0.83 CCNK (0.50) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL269583 0.83 CCNK (0.50) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL30259588 0.74 KDM4E (0.61) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL25258456 0.73 IDH2 (0.56) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL25222649 0.73 IDH2 (0.56) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL28312479 0.73 IDH2 (0.56) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL17961848 0.73 CCNT1 (0.41) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL17961847 0.73 CCNT1 (0.41) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL30833890 0.72 IDH2 (0.41) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL25294691 0.71 CCNT1 (0.41) CCNT1CCNKCDK9CDK12CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4347571-B1 TRIAZINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CANCER. HOFFMANN LA ROCHE (CH) 2026-04-22 EP disclosed
US-12421209-B2 Compounds HOFFMANN-LA ROCHE INC. (US) 2025-09-23 US disclosed
US-20250276958-A1 COMPOUNDS HOFFMANN-LA ROCHE INC. (US) 2025-09-04 US disclosed
US-20250197370-A1 NOVEL COMPOUNDS HOFFMANN-LA ROCHE INC. (US) 2025-06-19 US disclosed
US-20240132471-A1 NOVEL COMPOUNDS HOFFMANN-LA ROCHE INC. (US) 2024-04-25 US disclosed
EP-4347571-A1 TRIAZINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CANCER F. Hoffmann-La Roche AG (CH) 2024-04-10 EP disclosed
CN-117460718-A Triazine derivatives and their use in the treatment of cancer 豪夫迈·罗氏有限公司 2024-01-26 CN disclosed
WO-2022253936-A1 TRIAZINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CANCER. F. HOFFMANN-LA ROCHE AG (CH) 2022-12-08 WO disclosed
WO-2022253936-A1 TRIAZINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CANCER. F. HOFFMANN-LA ROCHE AG (CH) 2022-12-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12421209-B2 Compounds C5, RB1, RPS4X CCNT1 115/4885CCNK 311/4885CDK9 658/4885
US-20250276958-A1 COMPOUNDS C5, RB1, RPS4X CCNT1 115/4885CCNK 311/4885CDK9 658/4885
US-20250197370-A1 NOVEL COMPOUNDS RB1, CDK11B, RPS4X CCNT1 311/4885CCNK 484/4885CDK9 871/4885
US-20240132471-A1 NOVEL COMPOUNDS RB1, RPS4Y1, CDK11B CCNT1 294/4885CCNK 572/4885CDK9 842/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.