SCHEMBL24698462

SCHEMBL24698462

C[C@H]1CCN1c1nc2c(c(-c3cccc(S(N)(=O)=O)c3)n1)CCC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.42
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
LRRK2 Q5S007 1/20 0.37
PDE4D Q08499 1/20 0.37
PDE7A Q13946 1/20 0.37
TTK P33981 4/20 0.36
SYK P43405 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK8 P45983 2/20 0.35
ATR Q13535 1/20 0.35
ATRIP Q8WXE1 1/20 0.35
PIK3CD O00329 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015541 1.00 MTOR (0.42) MTORCA1CA2CA4CA7
SCHEMBL24698349 0.92 MTOR (0.36) MTORCYP1A2CYP2C19ATRATRIP
SCHEMBL30015473 0.92 MTOR (0.36) MTORCYP1A2CYP2C19ATRATRIP
SCHEMBL30015725 0.91 ATR (0.43) MTORCYP1A2CYP2C19ATRATRIP
SCHEMBL24697799 0.91 ATR (0.43) MTORCYP1A2CYP2C19ATRATRIP
SCHEMBL24698473 0.88 USP30 (0.41) MTORSYKMEN1KMT2A
SCHEMBL24698949 0.88 SYK (0.38) MTORSYKMAOACYP1A2CYP2C19
SCHEMBL24698105 0.87 HRH3 (0.40) CA1CA2CA7CA12CA9
SCHEMBL24699256 0.87 MEN1 (0.37) MTORCYP1A2CYP2C19ATRATRIP
SCHEMBL24697739 0.87 PIK3CD (0.35) MTORCYP2C19PIK3CDPIK3CAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed