SCHEMBL24698349

SCHEMBL24698349

C[C@H]1CCN1c1nc2c(c(-c3cccc(S(=N)(N)=O)c3)n1)CCC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.36
HRH3 Q9Y5N1 3/20 0.35
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
CYP2C19 P33261 2/20 0.34
CYP1A2 P05177 1/20 0.34
ATR Q13535 2/20 0.34
ATRIP Q8WXE1 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 4/20 0.33
HRH2 P25021 2/20 0.33
PIK3R1 P27986 4/20 0.33
PIK3CA P42336 4/20 0.33
GAA P10253 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015473 1.00 MTOR (0.36) MTORHRH3PDK1PDK2PDK3
SCHEMBL24698462 0.92 MTOR (0.42) MTORHRH3CYP2C19CYP1A2ATR
SCHEMBL30015541 0.92 MTOR (0.42) MTORHRH3CYP2C19CYP1A2ATR
SCHEMBL24699256 0.89 MEN1 (0.37) MTORHRH3PDK1PDK2PDK3
SCHEMBL24697799 0.89 ATR (0.43) MTORCYP2C19CYP1A2ATRATRIP
SCHEMBL30015725 0.89 ATR (0.43) MTORCYP2C19CYP1A2ATRATRIP
SCHEMBL24698930 0.88 ALDH1A1 (0.38) HRH3PDK1PDK2PDK3PDK4
SCHEMBL24698262 0.88 ATR (0.33) MTORHRH3PDK1PDK2PDK3
SCHEMBL24698949 0.86 SYK (0.38) MTORCYP2C19CYP1A2ATRATRIP
SCHEMBL24698473 0.86 USP30 (0.41) MTORMEN1KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed