SCHEMBL24698774

SCHEMBL24698774

C[C@H]1[C@H](F)CN1c1nc2c(c(-c3ccc(C(N)=O)cc3)n1)CCC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.35
HRH2 P25021 5/20 0.35
SMO Q99835 1/20 0.35
ALDH1A1 P00352 3/20 0.34
KDM1A O60341 1/20 0.34
KDM4E B2RXH2 2/20 0.33
CYP1A2 P05177 1/20 0.33
GAA P10253 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
HPGD P15428 2/20 0.32
MTOR P42345 1/20 0.32
EEF2K O00418 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
PDE2A O00408 1/20 0.32
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698766 1.00 HRH3 (0.35) HRH3HRH2SMOALDH1A1KDM1A
SCHEMBL24698714 0.89 HRH3 (0.36) HRH3HRH2SMOALDH1A1KDM1A
SCHEMBL24698818 0.89 HRH3 (0.36) HRH3HRH2SMOALDH1A1KDM1A
SCHEMBL24698712 0.89 HRH3 (0.36) HRH3HRH2SMOALDH1A1KDM1A
SCHEMBL24698713 0.89 HRH3 (0.36) HRH3HRH2SMOALDH1A1KDM1A
SCHEMBL24698716 0.89 HRH3 (0.36) HRH3HRH2SMOALDH1A1KDM1A
SCHEMBL24697597 0.88 HRH2 (0.36) HRH3HRH2SMOALDH1A1KDM1A
SCHEMBL24697789 0.88 ALDH1A1 (0.36) HRH3HRH2SMOALDH1A1KDM1A
SCHEMBL24698865 0.88 HRH2 (0.36) HRH3HRH2SMOALDH1A1KDM1A
SCHEMBL24698718 0.88 HRH3 (0.36) HRH3HRH2SMOALDH1A1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed