SCHEMBL24699080

SCHEMBL24699080

C[C@H]1CCN1c1nc2c(c(-c3cccc(S(=N)(=O)c4ccc(C#N)cc4)c3)n1)CCC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.39
HSD11B1 P28845 5/20 0.34
HRH3 Q9Y5N1 2/20 0.34
EGLN2 Q96KS0 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
CYP3A4 P08684 1/20 0.33
GRM5 P41594 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PTGS2 P35354 1/20 0.32
HTR6 P50406 1/20 0.32
PDK1 Q15118 1/20 0.32
PDK2 Q15119 1/20 0.32
PDK3 Q15120 1/20 0.32
PDK4 Q16654 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
CA1 P00915 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015974 1.00 TDP1 (0.39) TDP1HSD11B1HRH3EGLN2HTR2A
SCHEMBL24699256 0.90 MEN1 (0.37) HRH3SMN1; SMN2PDK1PDK2PDK3
SCHEMBL30014670 0.88 KCNK3 (0.34) TDP1HSD11B1EGLN2HTR2AHTR2C
SCHEMBL24697985 0.88 KCNK3 (0.34) TDP1HSD11B1EGLN2HTR2AHTR2C
SCHEMBL24699243 0.88 KDM1A (0.33) TDP1HRH3PDK1PDK2PDK3
SCHEMBL30016531 0.85 PI4KB (0.36) TDP1HRH3EGLN2HTR2AHTR2C
SCHEMBL24697976 0.85 PI4KB (0.36) TDP1HRH3EGLN2HTR2AHTR2C
SCHEMBL30015473 0.84 MTOR (0.36) HRH3PDK1PDK2PDK3PDK4
SCHEMBL24698349 0.84 MTOR (0.36) HRH3PDK1PDK2PDK3PDK4
SCHEMBL24698381 0.84 MTOR (0.41) HRH3CYP3A4TSHRSMN1; SMN2MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed