SCHEMBL24699338

SCHEMBL24699338

Cc1cc2c(N)n[nH]c2cn1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.53
GSK3B P49841 1/20 0.53
JAK2 O60674 11/20 0.44
PDPK1 O15530 6/20 0.44
UHRF1 Q96T88 1/20 0.42
DYRK1A Q13627 1/20 0.42
KDM4E B2RXH2 1/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
AURKA O14965 1/20 0.41
TGFBR1 P36897 1/20 0.41
ROCK1 Q13464 1/20 0.41
AURKB Q96GD4 1/20 0.41
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1640905 0.86 PDPK1 (0.46) GSK3AGSK3BJAK2PDPK1UHRF1
SCHEMBL7920977 0.82 ADORA2A (0.47) GSK3AGSK3BUHRF1DYRK1A
SCHEMBL15542652 0.79 JAK2 (0.40) GSK3AGSK3BJAK2UHRF1DYRK1A
SCHEMBL5826761 0.79 GSK3A (0.64) GSK3AGSK3BJAK2PDPK1AURKA
SCHEMBL12481324 0.78 PIM1 (0.33) GSK3AGSK3BUHRF1DYRK1A
SCHEMBL12479452 0.78 UHRF1 (0.36) GSK3AGSK3BJAK2PDPK1UHRF1
SCHEMBL31317680 0.78 UHRF1 (0.36) GSK3AGSK3BJAK2PDPK1UHRF1
SCHEMBL12480568 0.77 PRKAG1 (0.38) GSK3AGSK3BJAK2DYRK1AKDM4E
SCHEMBL16517125 0.77 PRKAG1 (0.47)
SCHEMBL17514104 0.76 JAK2 (0.53) GSK3AGSK3BJAK2PDPK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed