SCHEMBL24711535

SCHEMBL24711535

CNC(=O)N1CCN(C(C)C)C[C@@H]1C

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
HRH3 Q9Y5N1 5/20 0.33
SLC6A9 P48067 2/20 0.33
PRKCB P05771 1/20 0.33
MAPT P10636 1/20 0.32
CYP2D6 P10635 2/20 0.32
KCNH2 Q12809 1/20 0.32
IDH1 O75874 1/20 0.32
DRD4 P21917 1/20 0.31
LIMK2 P53671 2/20 0.31
GAA P10253 1/20 0.31
ROCK2 O75116 1/20 0.31
PRKG1 Q13976 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26240075 0.81 POLB (0.35) SMN1; SMN2POLBHRH3CYP2D6KCNH2
SCHEMBL26205553 0.81 SMN1; SMN2 (0.38) SMN1; SMN2TSHRHRH3SLC6A9PRKCB
SCHEMBL27157659 0.80 SMN1; SMN2 (0.40) SMN1; SMN2TSHRHRH3SLC6A9PRKCB
SCHEMBL16869402 0.80 SMN1; SMN2 (0.40) SMN1; SMN2POLBTSHRHRH3SLC6A9
SCHEMBL20008992 0.80 SMN1; SMN2 (0.40) SMN1; SMN2POLBTSHRHRH3SLC6A9
SCHEMBL20009022 0.80 SMN1; SMN2 (0.40) SMN1; SMN2POLBTSHRHRH3SLC6A9
SCHEMBL27204244 0.80 SMN1; SMN2 (0.40) SMN1; SMN2TSHRHRH3SLC6A9PRKCB
SCHEMBL24711925 0.79 TSHR (0.58) SMN1; SMN2TSHRHRH3SLC6A9PRKCB
SCHEMBL20008974 0.79 SMN1; SMN2 (0.41) SMN1; SMN2TSHRHRH3SLC6A9PRKCB
SCHEMBL23876806 0.79 PIK3CD (0.40) SMN1; SMN2TSHRHRH3SLC6A9PRKCB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230133671-A1 SETD2 INHIBITORS AND RELATED METHODS AND USES, INCLUDING COMBINATION THERAPIES Epizyme, Inc. (US) 2023-05-04 US disclosed
WO-2022261243-A1 COMBINATION THERAPIES WITH SETD2 INHIBITORS Epizyme, Inc. (US) 2022-12-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230133671-A1 SETD2 INHIBITORS AND RELATED METHODS AND USES, INCLUDING COMBINATION THERAPIES EZH2, HDAC2, SETD2 SMN1; SMN2 2240/4885POLB 2014/4885TSHR 2768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.