SCHEMBL2471646

SCHEMBL2471646

CNC(=O)c1c(-c2cc(C(=O)NC3(c4ccc5ncccc5n4)CC3)ccc2C)ccc2oc(-c3ccc(F)cc3)cc12

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.62
CYP3A4 P08684 5/20 0.62
KCNH2 Q12809 3/20 0.62
NR1I2 O75469 1/20 0.62
MAPK14 Q16539 1/20 0.35
IDO1 P14902 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL120717 0.88 CYP2C8 (0.79) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL2471972 0.88 CYP2C8 (0.58) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL121622 0.87 CYP2C8 (0.79) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL2471645 0.85 CYP2C8 (0.57) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL146317 0.79 CYP2C8 (0.79) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL120739 0.78 CYP2C8 (0.65) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL139473 0.77 CYP2C8 (0.79) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL2141972 0.76 CYP2C8 (1.00) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL145125 0.76 CYP2C8 (0.75) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL143691 0.76 CYP2C8 (0.75) CYP2C8CYP3A4KCNH2NR1I2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545051-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112769-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed