SCHEMBL24718682

SCHEMBL24718682

CCOC(=O)c1ccc(Br)c(Cl)c1CBr

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.51
CYP4A11 Q02928 1/20 0.51
TSHR P16473 1/20 0.46
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
CA12 O43570 3/20 0.43
CA9 Q16790 3/20 0.43
CA7 P43166 2/20 0.43
CA14 Q9ULX7 2/20 0.43
PLK1 P53350 1/20 0.42
MAOB P27338 1/20 0.41
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 1/20 0.41
KDM4E B2RXH2 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
MAPK1 P28482 1/20 0.39
METTL3 Q86U44 1/20 0.39
BAZ2B Q9UIF8 1/20 0.38
BAZ2A Q9UIF9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7573933 0.86 CYP4F2 (0.60) CYP4F2CYP4A11TSHRCA1CA2
SCHEMBL18786802 0.84 ABL1 (0.41) TSHRCA1CA2CA12CA9
SCHEMBL30798535 0.83 TSHR (0.50) CYP4F2CYP4A11TSHRCA1CA2
SCHEMBL24718020 0.83 TSHR (0.50) CYP4F2CYP4A11TSHRCA1CA2
SCHEMBL7523025 0.83 TSHR (0.50) CYP4F2CYP4A11TSHRCA1CA2
SCHEMBL8729880 0.82 CYP4F2 (0.58) CYP4F2CYP4A11TSHRCA1CA2
SCHEMBL8724253 0.78 TSHR (0.58) CYP4F2CYP4A11TSHRCA1CA2
SCHEMBL30772831 0.78 TSHR (0.58) CYP4F2CYP4A11TSHRCA1CA2
SCHEMBL2601357 0.77 CYP4F2 (0.56) CYP4F2CYP4A11TSHRCA1CA2
SCHEMBL27797134 0.76 TSHR (0.59) CYP4F2CYP4A11TSHRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220395576-A1 MODULATORS OF BCL6 PROTEOLYSIS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. 2022-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220395576-A1 MODULATORS OF BCL6 PROTEOLYSIS AND ASSOCIATED METHODS OF USE BCL6, BCL6B, BCL3 CYP4F2 4269/4885CYP4A11 4137/4885TSHR 3100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.