SCHEMBL24719019

SCHEMBL24719019

O=C1c2ccccc2C(=O)N1Cc1ccc(Cl)nn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
MEN1 O00255 1/20 0.54
PKM P14618 1/20 0.54
KMT2A Q03164 1/20 0.54
TYR P14679 4/20 0.51
MAPT P10636 2/20 0.48
RECQL P46063 2/20 0.48
CASP3 P42574 2/20 0.47
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
GLS O94925 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
KDM4E B2RXH2 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30146401 1.00 ALDH1A1 (0.54) ALDH1A1MEN1PKMKMT2ATYR
SCHEMBL241916 0.75 ALDH1A1 (0.65) ALDH1A1MEN1PKMKMT2ATYR
SCHEMBL29411233 0.74 MEN1 (0.55) ALDH1A1MEN1PKMKMT2ATYR
SCHEMBL29411247 0.74 ALDH1A1 (0.51) ALDH1A1MEN1PKMKMT2ATYR
SCHEMBL17979341 0.74 MEN1 (0.55) ALDH1A1MEN1PKMKMT2ATYR
SCHEMBL3720990 0.74 ALDH1A1 (0.51) ALDH1A1MEN1PKMKMT2ATYR
SCHEMBL17979249 0.74 ALDH1A1 (0.51) ALDH1A1MEN1PKMKMT2ATYR
SCHEMBL29411219 0.74 ALDH1A1 (0.51) ALDH1A1MEN1PKMKMT2ATYR
SCHEMBL21555613 0.74 TYR (0.46) ALDH1A1MEN1PKMKMT2ATYR
SCHEMBL8218007 0.74 ALDH1A1 (0.51) ALDH1A1MEN1PKMKMT2ATYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117412973-A Nitrogen-containing fused heteroaromatic bicyclic compounds as USP1 inhibitors and uses thereof 上海瑛派药业有限公司 2024-01-16 CN disclosed
WO-2022253188-A1 NITROGEN-CONTAINING FUSED HETEROAROMATIC BICYCLIC COMPOUNDS AS USP1 INHIBITORS AND THE USE THEREOF IMPACT THERAPEUTICS (SHANGHAI) , INC (CN) 2022-12-08 WO disclosed