SCHEMBL24722714

SCHEMBL24722714

CC(C)(C)NC1Cc2cc(Br)cnc2NC1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.34
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
NNMT P40261 1/20 0.32
BRD4 O60885 1/20 0.31
AURKA O14965 1/20 0.31
DAPK3 O43293 1/20 0.31
JAK2 O60674 1/20 0.31
PRKD3 O94806 1/20 0.31
MAP4K4 O95819 1/20 0.31
PAK4 O96013 1/20 0.31
ABL1 P00519 1/20 0.31
NTRK1 P04629 1/20 0.31
FYN P06241 1/20 0.31
RET P07949 1/20 0.31
MET P08581 1/20 0.31
PDGFRB P09619 1/20 0.31
PIM1 P11309 1/20 0.31
FGFR1 P11362 1/20 0.31
PDGFRA P16234 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21366217 0.81 GAA (0.43) DDB1CRBNNNMT
SCHEMBL29799886 0.81 GAA (0.43) DDB1CRBNNNMT
SCHEMBL21358706 0.79 SMYD3 (0.36) NNMTAURKADAPK3JAK2PRKD3
SCHEMBL24722621 0.78 KDM4E (0.32)
SCHEMBL2276398 0.77 AKR1B1 (0.40) AKR1B1DDB1CRBNNNMTBRD4
SCHEMBL726486 0.75 NNMT (0.36) AKR1B1NNMT
SCHEMBL30304181 0.75 CRBN (0.37) AKR1B1DDB1CRBNAURKADAPK3
SCHEMBL24823109 0.75 CRBN (0.37) AKR1B1DDB1CRBNAURKADAPK3
SCHEMBL2672662 0.74 NNMT (0.36) AKR1B1CRBNNNMTAURKADAPK3
SCHEMBL23554694 0.73 GAA (0.41) DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022187329-A1 FABI INHIBITORS FOR GRAM-NEGATIVE PATHOGENS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2022-09-09 WO disclosed