SCHEMBL24726652

SCHEMBL24726652

CC(C)c1cccc(-c2ccc3ncnn3c2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.51
TGFBR1 P36897 4/20 0.48
MAPK14 Q16539 1/20 0.48
SCN5A Q14524 1/20 0.45
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
RXRG P48443 1/20 0.42
TLR9 Q9NR96 4/20 0.42
TLR8 Q9NR97 4/20 0.42
TLR7 Q9NYK1 4/20 0.42
PIK3CD O00329 1/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
JAK2 O60674 1/20 0.40
PTPN5 P54829 2/20 0.40
NR4A2 P43354 1/20 0.40
ABL1 P00519 1/20 0.38
SRC P12931 1/20 0.38
TNIK Q9UKE5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24726642 0.81 MAPK1 (0.41) TGFBR1MAPK14RXRARXRBRXRG
SCHEMBL12609895 0.76 DYRK1A (0.60) DYRK1ATGFBR1MAPK14SCN5APIK3CD
SCHEMBL84387 0.76 DYRK1A (0.44) DYRK1ATGFBR1MAPK14SCN5ATLR9
SCHEMBL30014450 0.74 DYRK1A (0.51) DYRK1ATGFBR1MAPK14SCN5APIK3CD
SCHEMBL30013771 0.74 EGLN2 (0.58) DYRK1ATGFBR1MAPK14SCN5A
SCHEMBL749404 0.74 DYRK1A (0.51) DYRK1ATGFBR1MAPK14SCN5APIK3CD
SCHEMBL938164 0.73 DYRK1A (0.50) DYRK1ATGFBR1MAPK14SCN5APIK3CD
SCHEMBL30013812 0.72 DYRK1A (0.49) DYRK1ATGFBR1MAPK14SCN5APIK3CD
SCHEMBL30014288 0.72 DYRK1A (0.49) DYRK1ATGFBR1MAPK14SCN5APIK3CD
SCHEMBL5352034 0.72 RXRA (0.62) RXRARXRBRXRGPTPN5NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234965-A1 HETEROARYL DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT 주식회사 보로노이 2022-11-10 WO disclosed