SCHEMBL24735358

SCHEMBL24735358

Bc1c(B)c(B)c2c(-c3cccc4oc5c6ccccc6ccc5c34)c3c(B)c(B)c(B)c(B)c3c(-c3ccc(-c4ccccc4)c(-c4ccccc4)c3)c2c1B

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 12/20 0.37
CYP1B1 Q16678 12/20 0.37
CYP1A2 P05177 11/20 0.37
ABCG2 Q9UNQ0 3/20 0.37
PRKDC P78527 3/20 0.37
ABCC1 P33527 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
PDE5A O76074 1/20 0.37
TP53 P04637 1/20 0.37
ABCB1 P08183 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP19A1 P11511 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
CYP2B6 P20813 1/20 0.37
TACR2 P21452 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22382184 0.90 CYP1A1 (0.39) CYP1A1CYP1B1CYP1A2ABCG2PRKDC
SCHEMBL21940072 0.90 CYP1A1 (0.39) CYP1A1CYP1B1CYP1A2ABCG2PRKDC
SCHEMBL22541952 0.88 CYP1A1 (0.40) CYP1A1CYP1B1CYP1A2ABCG2PRKDC
SCHEMBL24859961 0.85 CYP1A1 (0.33) CYP1A1CYP1B1CYP1A2ABCG2PRKDC
SCHEMBL24908328 0.85 CYP1A1 (0.37) CYP1A1CYP1B1CYP1A2ABCG2PRKDC
SCHEMBL24766722 0.85 CYP1A1 (0.42) CYP1A1CYP1B1CYP1A2ABCG2PRKDC
SCHEMBL26591896 0.84 ARSA (0.38) CYP1A1CYP1B1CYP1A2ABCG2PRKDC
SCHEMBL24469249 0.84 CYP1A1 (0.36) CYP1A1CYP1B1CYP1A2ABCG2PRKDC
SCHEMBL23109579 0.84 ALDH1A1 (0.32) ALDH1A1MAPTKDM4E
SCHEMBL24481438 0.83 ARSA (0.34) CYP1A1CYP1B1CYP1A2ABCG2PRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220393110-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT, COMPOSITION, POWDER, ELECTRONIC EQUIPMENT, AND NOVEL COMPOUND IDEMITSU KOSAN CO.,LTD. (CN) 2022-12-08 US disclosed