SCHEMBL247361

SCHEMBL247361

CCCCCOc1ccc(C(=O)c2cccc3ccccc23)c2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 17/20 1.00
CNR1 P21554 12/20 1.00
CYP2C9 P11712 1/20 1.00
THRA P10827 1/20 0.58
THRB P10828 1/20 0.58
MEN1 O00255 1/20 0.57
HTT P42858 1/20 0.57
KMT2A Q03164 1/20 0.57
CDC25B P30305 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29362406 1.00 CNR2 (1.00) CNR2CNR1CYP2C9THRATHRB
Naphthoic Acid SCHEMBL27493013 0.95 CNR2 (0.91) CNR2CNR1CYP2C9THRATHRB
SCHEMBL247971 0.90 CNR2 (0.80) CNR2CNR1CYP2C9THRATHRB
SCHEMBL247905 0.87 CNR2 (0.77) CNR2CNR1CYP2C9THRATHRB
SCHEMBL15995238 0.87 CNR2 (0.79) CNR2CNR1CYP2C9THRATHRB
SCHEMBL27493012 0.86 CNR2 (0.75) CNR2CNR1CYP2C9MEN1KMT2A
SCHEMBL250281 0.86 CNR2 (0.74) CNR2CNR1CYP2C9THRATHRB
SCHEMBL248582 0.86 CNR2 (0.74) CNR2CNR1CYP2C9THRATHRB
SCHEMBL249236 0.86 CNR2 (0.74) CNR2CNR1CYP2C9THRATHRB
SCHEMBL27557505 0.86 CNR2 (0.74) CNR2CNR1CYP2C9MEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 87 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170014355-A1 CANNABINOID RECEPTOR TREATMENTS TEMPLE UNIVERSITY OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2017-01-19 US claimed
WO-2013025984-A2 CANNABINOID RECEPTOR TREATMENTS TEMPLE UNIVERSITY (US) 2013-02-21 WO claimed
EP-1339663-B1 NAPHTHALENE DERIVATIVES NOVARTIS AG (CH) 2012-01-04 EP claimed
EP-2305215-A1 Microemulsions of cannabinoid receptor binding compounds Novartis AG (CH) 2011-04-06 EP claimed
US-7763607-B2 Pharmaceutical compositions comprising CBx cannabinoid receptor modulators and potassium channel modulators SOLVAY PHARMACEUTICALS GMBH (DE) 2010-07-27 US claimed
EP-2065033-A1 Microemulsions of cannabinoid receptor binding compounds Novartis Ag (CH) 2009-06-03 EP claimed
US-20080279940-A1 Microemulsions of Cannabinoid Receptor Binding Compounds NOVARTIS AG (CH) 2008-11-13 US claimed
WO-2008033351-A2 MULTIMODAL ABUSE RESISTANT AND EXTENDED RELEASE FORMULATIONS THERAQUEST BIOSCIENCES, INC. (US) 2008-03-20 WO claimed
WO-2008024490-A2 ORAL PHARMACEUTICAL FORMULATIONS OF ABUSE DETERRENT CANNABINOIDS AND METHOD OF USE THERAQUEST BIOSCIENCES, INC. (US) 2008-02-28 WO claimed
EP-1858484-A1 MICROEMULSIONS OF CANNABINOID RECEPTOR BINDING COMPOUNDS Novartis AG (CH) 2007-11-28 EP claimed
WO-2006094829-A1 MICROEMULSIONS OF CANNABINOID RECEPTOR BINDING COMPOUNDS NOVARTIS AG (CH) 2006-09-14 WO claimed
US-20240082270-A1 CANNABIGEROL (CBG) PRODUCTS AND METHODS OF USE BAZELET HEALTH SYSTEMS INC (US) 2024-03-14 US disclosed
US-20210121414-A1 METHOD FOR PRODUCING A PHARMACEUTICAL COMPOSITION OF POLYMERIC NANOPARTICLES FOR TREATING NEUROPATHIC PAIN CAUSED BY PERIPHERAL NERVE COMPRESSION UNIV SEVILLA (ES) 2021-04-29 US disclosed
EP-2744778-B1 META-SUBSTITUTED BIPHENYL PERIPHERALLY RESTRICTED FAAH INHIBITORS UNIV CALIFORNIA (US) 2019-01-16 EP disclosed
US-20180200225-A1 HYDRAZONE MODULATORS OF CANNABINOID RECEPTORS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2018-07-19 US disclosed
US-7045533-B2 Such as naphthalen-1-yl-(4-pentyloxy-naphthalen-1-yl)-mehtane for treatment/prevention of diseases/conditions associated with cannobinoid receptor activation such as chronic pain, osteo- and rheumatoid arthritis, teno-synovitis and gout NOVARTIS AG (CH) 2006-05-16 US disclosed
WO-2005058292-A1 NEW USE IN GASTROINTESTINAL DISORDERS ASTRAZENECA AB (SE) 2005-06-30 WO disclosed
US-20040053890-A1 Naphthalene derivatives NOVARTIS AG (CH) 2004-03-18 US disclosed
EP-1339663-A2 NAPHTHALENE DERIVATIVES Novartis AG (CH) 2003-09-03 EP disclosed
WO-2002042248-A2 NAPHTHALENE DERIVATIVES NOVARTIS AG (CH) 2002-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170014355-A1 CANNABINOID RECEPTOR TREATMENTS CNR1, CNR2, GPR18 CNR2 2/4885CNR1 1/4885CYP2C9 786/4885
US-20080279940-A1 Microemulsions of Cannabinoid Receptor Binding Compounds CNR1, CNR2, OPRL1 CNR2 2/4885CNR1 1/4885CYP2C9 1204/4885
US-20040053890-A1 Naphthalene derivatives CYP1A1, SULT1E1, CYP2F1 CNR2 86/4885CNR1 35/4885CYP2C9 149/4885
US-20180200225-A1 HYDRAZONE MODULATORS OF CANNABINOID RECEPTORS CNR1, CNR2, GPR18 CNR2 2/4885CNR1 1/4885CYP2C9 743/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.