SCHEMBL2474337

SCHEMBL2474337

CC(C)(C)OC(=O)N1Cc2ccccc2-n2cnnc2C1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.46
NAMPT P43490 4/20 0.43
ESR2 Q92731 1/20 0.42
NR1H2 P55055 2/20 0.40
SMARCA2 P51531 1/20 0.40
SMARCA4 P51532 1/20 0.40
PBRM1 Q86U86 1/20 0.40
DDB1 Q16531 2/20 0.39
CRBN Q96SW2 2/20 0.39
BCHE P06276 1/20 0.39
HDAC1 Q13547 1/20 0.38
GRM5 P41594 1/20 0.37
GRM1 Q13255 1/20 0.37
NOTUM Q6P988 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2328281 0.84 AVPR1A (0.49) ESR2NR1H2
SCHEMBL3765031 0.84 ESR2 (0.41) MAPK1ESR2NR1H2DDB1CRBN
SCHEMBL3762487 0.81 MAPK1 (0.49) MAPK1NAMPTESR2NR1H2DDB1
SCHEMBL2578140 0.78 TACR1 (0.34) MAPK1NAMPTESR2NR1H2SMARCA2
SCHEMBL12197348 0.78 MAPK1 (0.46) MAPK1NAMPTESR2NR1H2DDB1
SCHEMBL29676965 0.77 MAPK1 (0.64) MAPK1NAMPTESR2NR1H2DDB1
SCHEMBL5183098 0.77 MAPK1 (0.64) MAPK1NAMPTESR2NR1H2DDB1
SCHEMBL2550063 0.77 NAMPT (0.40) NAMPTESR2DDB1CRBN
SCHEMBL2573980 0.76 DDB1 (0.38) MAPK1ESR2NR1H2SMARCA2SMARCA4
SCHEMBL2478651 0.75 USP30 (0.37) DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250157-B1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LTD (IN) 2014-11-05 EP disclosed
EP-2370441-A1 ARYLCYCLOHEXYLETHERS OF DIHYDROTETRAAZABENZOAZULENES FOR USE AS VASOPRESSIN VIA RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2011-10-05 EP disclosed