SCHEMBL2550063

SCHEMBL2550063

CC(C)(C)OC(=O)N1Cc2cc(C3(Cl)CCC(c4ccccc4)CC3)ccc2-n2cnnc2C1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.40
DDB1 Q16531 2/20 0.37
CRBN Q96SW2 2/20 0.37
AVPR1A P37288 2/20 0.37
OXTR P30559 1/20 0.37
RORC P51449 2/20 0.36
TP53 P04637 3/20 0.34
GPR119 Q8TDV5 2/20 0.34
MAPT P10636 1/20 0.34
TACR1 P25103 1/20 0.34
LMNA P02545 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
USP30 Q70CQ3 1/20 0.33
ESR2 Q92731 1/20 0.33
AVPR2 P30518 1/20 0.33
KCNH2 Q12809 1/20 0.33
KDM1A O60341 1/20 0.33
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2556747 0.91 HDAC1 (0.38) NAMPTDDB1CRBNAVPR1AOXTR
SCHEMBL2579657 0.90 OXTR (0.36) DDB1CRBNAVPR1AOXTRGPR119
SCHEMBL2565904 0.90 AVPR2 (0.37) NAMPTDDB1CRBNAVPR1AOXTR
SCHEMBL2552066 0.89 GPR119 (0.38) NAMPTDDB1CRBNAVPR1AOXTR
SCHEMBL2549514 0.89 MGLL (0.35) NAMPTDDB1CRBNAVPR1AOXTR
SCHEMBL2580027 0.88 DDB1 (0.36) DDB1CRBNAVPR1AOXTRGPR119
SCHEMBL2578140 0.88 TACR1 (0.34) NAMPTDDB1CRBNAVPR1AOXTR
SCHEMBL2565485 0.88 FNTA (0.37) DDB1CRBNAVPR1AOXTRGPR119
SCHEMBL2574746 0.88 OXTR (0.34) NAMPTDDB1CRBNAVPR1AOXTR
SCHEMBL2580300 0.88 OXTR (0.36) DDB1CRBNAVPR1AOXTRGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552919-A1 ARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. Hoffmann-La Roche AG (CH) 2013-02-06 EP disclosed
WO-2011120877-A1 ARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-06 WO disclosed