SCHEMBL24757337

SCHEMBL24757337

Cc1c(C(C)(F)F)nn(C[C@H]2CCC(F)(F)C2)c1C(=O)Nc1cccc(SN)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
ANO1 Q5XXA6 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
KIF18A Q8NI77 2/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ACKR3 P25106 4/20 0.32
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
FLT1 P17948 1/20 0.31
KDR P35968 1/20 0.31
TRPV4 Q9HBA0 1/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24757338 1.00 AKR1C3 (0.39) AKR1C3AKR1C2ANO1CHRM2CHRM1
SCHEMBL24906338 0.87 SCN10A (0.43) AKR1C3AKR1C2KIF18AALDH1A1MEN1
SCHEMBL24906520 0.87 SCN10A (0.43) AKR1C3AKR1C2KIF18AALDH1A1MEN1
SCHEMBL24906523 0.87 SCN10A (0.43) AKR1C3AKR1C2KIF18AALDH1A1MEN1
SCHEMBL24757786 0.84 ANO1 (0.44) AKR1C3AKR1C2ANO1
SCHEMBL30141516 0.82 ANO1 (0.40) AKR1C3AKR1C2ANO1
SCHEMBL24757840 0.82 AKR1C3 (0.40) AKR1C3AKR1C2CHRM2CHRM1CHRM3
SCHEMBL24906478 0.81 SCN10A (0.48)
SCHEMBL24906419 0.81 SCN10A (0.45) AKR1C3AKR1C2MEN1KMT2A
SCHEMBL24758438 0.81 ANO1 (0.38) AKR1C3AKR1C2ANO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022263498-A1 SUBSTITUTED PYRAZOLE AMIDES Grünenthal GmbH (DE) 2022-12-22 WO disclosed