SCHEMBL24763592

SCHEMBL24763592

CC(C)(C)OC(=O)N1CCN(c2cnc(C(F)(F)F)cn2)C(CO)C1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
GPR119 Q8TDV5 15/20 0.43
CKS1B P61024 1/20 0.38
SKP1 P63208 1/20 0.38
SKP2 Q13309 1/20 0.38
NR1H2 P55055 2/20 0.38
NR1H3 Q13133 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26959278 1.00 HDAC8 (0.43) HDAC8HDAC6GPR119CKS1BSKP1
SCHEMBL24675569 1.00 HDAC8 (0.43) HDAC8HDAC6GPR119CKS1BSKP1
SCHEMBL28966515 0.86 GPR119 (0.51) HDAC8HDAC6GPR119CKS1BSKP1
SCHEMBL28966512 0.86 GPR119 (0.51) HDAC8HDAC6GPR119CKS1BSKP1
SCHEMBL29841788 0.85 HDAC6 (0.46) HDAC8HDAC6GPR119CKS1BSKP1
SCHEMBL26915117 0.85 HDAC6 (0.46) HDAC8HDAC6GPR119CKS1BSKP1
SCHEMBL29088932 0.85 HDAC6 (0.46) HDAC8HDAC6GPR119CKS1BSKP1
SCHEMBL26915035 0.85 CHRM2 (0.40) NR1H2NR1H3
SCHEMBL29274283 0.85 CHRM2 (0.40) NR1H2NR1H3
SCHEMBL21360407 0.84 GPR119 (0.56) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117083274-A Fused ring heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2023-11-17 CN disclosed
CN-116724044-A Tri-heterocyclic compound, preparation method and application thereof 上海湃隆生物科技有限公司 2023-09-08 CN disclosed
WO-2022184103-A1 TRICYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 武汉誉祥医药科技有限公司 2022-09-09 WO disclosed