SCHEMBL24765640

SCHEMBL24765640

CCC(N)Cc1cc(OC)c(C(F)(F)OC)cc1OC

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.46
HTR2C P28335 2/20 0.46
TAAR1 Q96RJ0 3/20 0.45
HTR1A P08908 1/20 0.43
HTR2B P41595 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24765901 1.00 HTR2A (0.46) HTR2AHTR2CTAAR1HTR1AHTR2B
SCHEMBL24765861 0.92 HTR2A (0.39) HTR2AHTR2CTAAR1HTR1AHTR2B
SCHEMBL24765870 0.92 TAAR1 (0.41) HTR2AHTR2CTAAR1HTR1AHTR2B
SCHEMBL24765899 0.88 HTR2A (0.59) HTR2AHTR2CTAAR1
SCHEMBL24765639 0.88 HTR2A (0.59) HTR2AHTR2CTAAR1
SCHEMBL24765644 0.87 HTR2A (0.47) HTR2AHTR2CTAAR1
SCHEMBL24765863 0.86 HTR2A (0.34) HTR2AHTR2CTAAR1HTR1AHTR2B
SCHEMBL24765654 0.81 HTR2A (0.50) HTR2AHTR2CTAAR1
SCHEMBL24765647 0.81 HTR2A (0.50) HTR2AHTR2CTAAR1
SCHEMBL30855223 0.79 TAAR1 (0.47) HTR2ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022204323-A1 NON-HALLUCINOGENIC ARIADNE ANALOGS FOR TREATMENT OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2022-09-29 WO disclosed