SCHEMBL2476644

SCHEMBL2476644

CN(Cc1ccccc1Cl)C(=O)[C@@]1(c2ccccc2)C[C@H]1CO

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 8/20 0.55
SLC6A2 P23975 8/20 0.54
SLC6A4 P31645 6/20 0.54
SLC6A3 Q01959 5/20 0.54
CYP2D6 P10635 1/20 0.46
HTR2C P28335 1/20 0.46
KDM4E B2RXH2 1/20 0.45
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2480415 0.93 TACR3 (0.51) TACR3SLC6A2SLC6A4SLC6A3
SCHEMBL2478849 0.91 TACR3 (0.51) TACR3SLC6A2SLC6A4SLC6A3
SCHEMBL2482572 0.89 TACR3 (0.63) TACR3
SCHEMBL2478511 0.86 TACR3 (0.51) TACR3
SCHEMBL2480492 0.85 SLC6A2 (0.59) TACR3SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL2477546 0.82 TACR3 (0.55) TACR3SLC6A2SLC6A4SLC6A3
SCHEMBL2480969 0.80 TACR3 (0.62) TACR3SLC6A2SLC6A4SLC6A3
SCHEMBL2477184 0.79 TACR3 (0.65) TACR3
SCHEMBL2478297 0.77 TACR3 (0.67) TACR3
SCHEMBL2479387 0.77 TACR3 (0.67) TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656349-B1 CYCLOPROPYL DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS LUNDBECK & CO AS H (DK) 2011-10-12 EP disclosed