SCHEMBL24767919

SCHEMBL24767919

Clc1ccc2ncnc(Nc3ccc(Cc4ccn5ncnc5c4)cc3)c2n1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.47
MKNK2 Q9HBH9 8/20 0.42
NTRK1 P04629 1/20 0.37
ERBB2 P04626 1/20 0.36
NQO2 P16083 1/20 0.36
FECH P22830 1/20 0.36
MYH14 Q7Z406 1/20 0.36
RIPK3 Q9Y572 1/20 0.36
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
GLA P06280 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30575827 0.87 EGFR (0.45) EGFRMKNK2ERBB2NQO2FECH
SCHEMBL25430634 0.87 EGFR (0.45) EGFRMKNK2ERBB2NQO2FECH
SCHEMBL30127392 0.82 EGFR (0.47) EGFRMKNK2ERBB2NQO2FECH
SCHEMBL30127072 0.82 EGFR (0.47) EGFRMKNK2ERBB2NQO2FECH
SCHEMBL24167293 0.80 EGFR (0.52) EGFRERBB2NQO2FECHMYH14
SCHEMBL24569376 0.80 KDM4E (0.53) EGFRERBB2NQO2FECHMYH14
SCHEMBL29888339 0.80 KDM4E (0.53) EGFRERBB2NQO2FECHMYH14
SCHEMBL24569439 0.76 ERBB2 (0.61) EGFRERBB2NQO2FECHMYH14
SCHEMBL29888106 0.76 ERBB2 (0.61) EGFRERBB2NQO2FECHMYH14
SCHEMBL29887854 0.76 ERBB2 (0.61) EGFRERBB2NQO2FECHMYH14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022266458-A1 6-HETEROCYCLOALKYL-QUINAZOLINE DERIVATIVES AND USES THEREOF BLACK DIAMOND THERAPEUTICS, INC. (US) 2022-12-22 WO disclosed