SCHEMBL24767970

SCHEMBL24767970

Bc1ccc(C)nc1C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
S1PR4 O95977 1/20 0.32
GRM6 O15303 1/20 0.32
GRM5 P41594 3/20 0.32
HPGDS O60760 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17281237 0.83 CNR1 (0.39) ALDH1A1LMNACNR1CNR2CYP2C9
SCHEMBL29202717 0.80 CNR1 (0.37) ALDH1A1LMNACNR1CNR2CYP2C9
SCHEMBL30322363 0.80 CNR1 (0.37) ALDH1A1LMNACNR1CNR2CYP2C9
SCHEMBL14634345 0.80 GRM5 (0.47) ALDH1A1LMNACNR1CNR2CYP2C9
SCHEMBL28593194 0.72 S1PR4 (0.40) ALDH1A1LMNACNR1CNR2S1PR4
SCHEMBL23345398 0.70 EGFR (0.43) ALDH1A1LMNACNR1CNR2
SCHEMBL946380 0.69 P2RX7 (0.50) ALDH1A1CYP2C9CYP2C19GRM5HPGDS
SCHEMBL32315381 0.69 P2RX7 (0.50) ALDH1A1CYP2C9CYP2C19GRM5HPGDS
SCHEMBL22866604 0.69 CNR1 (0.44) ALDH1A1LMNACNR1CNR2CYP2C9
SCHEMBL264062 0.68 ATR (0.44) NPSR1S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4104865-A1 ANTI-EGFR ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2022-12-21 EP disclosed