SCHEMBL2477358

SCHEMBL2477358

CC(=O)NC1(c2ccccc2)CCN(C[C@@H]2C[C@@H]2c2ccc(F)c(F)c2)CC1.CC(c1ccccc1)N(C)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 17/20 0.50
TACR2 P21452 3/20 0.42
TACR1 P25103 2/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2478061 0.89 TACR2 (0.53) TACR3TACR2TACR1
SCHEMBL2477155 0.89 TACR2 (0.53) TACR3TACR2TACR1
SCHEMBL2481967 0.83 TACR3 (0.56) TACR3TACR2TACR1
SCHEMBL2480824 0.82 TACR3 (0.57) TACR3TACR2TACR1
SCHEMBL2504727 0.80 CCR5 (0.39) TACR3TACR2TACR1CYP2C19
SCHEMBL2479278 0.78 TACR3 (0.71) TACR3TACR2TACR1
SCHEMBL2476101 0.78 TACR3 (0.71) TACR3TACR2TACR1
SCHEMBL2479040 0.77 TACR3 (0.51) TACR3TACR2TACR1CYP2C19
SCHEMBL2482748 0.77 TACR3 (0.51) TACR3TACR2TACR1CYP2C19
SCHEMBL2477495 0.76 TACR3 (0.66) TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656349-B1 CYCLOPROPYL DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS LUNDBECK & CO AS H (DK) 2011-10-12 EP claimed