SCHEMBL24775286

SCHEMBL24775286

C=C1CC(C=O)(c2ccc(Br)cc2)C1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.32
CYP2A6 P11509 1/20 0.31
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30
PIM1 P11309 1/20 0.30
PIM2 Q9P1W9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13307802 0.80 EGFR (0.35) CYP2A6MAOAMAOB
SCHEMBL4046273 0.79 CYP2A6 (0.36) CYP2A6MAOAMAOBPIM1PIM2
SCHEMBL20582009 0.76 LIG1 (0.41) CYP2A6MAOAMAOBPIM1PIM2
SCHEMBL4770412 0.76 LIG1 (0.37) CYP2A6MAOAMAOBPIM1PIM2
SCHEMBL14710732 0.74 TAAR1 (0.35) CNR1CYP2A6MAOAMAOBPIM1
SCHEMBL28937814 0.72 LIG1 (0.34)
SCHEMBL28173283 0.72 MMP2 (0.35) MAOAMAOBPIM1PIM2
Hydrochloric Acid SCHEMBL28028597 0.70 MMP2 (0.35) MAOAMAOBPIM1PIM2
SCHEMBL21944284 0.67 MMP2 (0.33)
SCHEMBL31219459 0.67 CYP2A6 (0.36) CNR1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022257961-A1 BENZOHETEROCYCLIC COMPOUND FOR TREATING EP2 AND EP4 RECEPTOR-MEDIATED DISEASES 武汉人福创新药物研发中心有限公司 2022-12-15 WO disclosed
CN-115448882-A Benzoheterocyclic compounds useful for the treatment of EP2, EP4 receptor mediated diseases 武汉人福创新药物研发中心有限公司 2022-12-09 CN disclosed