SCHEMBL2478285

SCHEMBL2478285

C[C@@H](c1ccccc1)N(C)C(=O)O.O=C(N1CCCCC1)C1(c2ccccc2)CCN(C[C@@H]2C[C@@H]2c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 4/20 0.54
HSD11B1 P28845 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DRD2 P14416 2/20 0.38
DRD4 P21917 2/20 0.38
NPY1R P25929 2/20 0.38
TACR2 P21452 5/20 0.38
TACR1 P25103 3/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SLC6A4 P31645 1/20 0.37
KCNH2 Q12809 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2477401 0.88 TACR3 (0.44) TACR3HSD11B1MEN1KMT2ADRD2
SCHEMBL2480350 0.87 TACR3 (0.67) TACR3HSD11B1MEN1KMT2ATACR2
SCHEMBL2477412 0.85 TACR3 (0.60) TACR3HSD11B1TACR2TACR1
SCHEMBL2479040 0.84 TACR3 (0.51) TACR3DRD2DRD4TACR2TACR1
SCHEMBL2482748 0.84 TACR3 (0.51) TACR3DRD2DRD4TACR2TACR1
SCHEMBL2477155 0.84 TACR2 (0.53) TACR3TACR2TACR1
SCHEMBL2478061 0.84 TACR2 (0.53) TACR3TACR2TACR1
SCHEMBL2476377 0.80 TACR3 (0.75) TACR3TACR2TACR1
SCHEMBL2480965 0.80 TACR3 (0.75) TACR3TACR2TACR1
SCHEMBL2477355 0.80 TACR3 (0.75) TACR3TACR2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656349-B1 CYCLOPROPYL DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS LUNDBECK & CO AS H (DK) 2011-10-12 EP claimed