SCHEMBL2478377

SCHEMBL2478377

O=C(Nc1ccc(Oc2ccnc(C(=O)NCO)c2)cc1)Nc1ccc(Br)c(C(F)(F)F)c1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 13/20 0.86
KDR P35968 3/20 0.66
HDAC3 O15379 6/20 0.65
HDAC4 P56524 6/20 0.65
HDAC1 Q13547 6/20 0.65
HDAC7 Q8WUI4 6/20 0.65
HDAC2 Q92769 6/20 0.65
HDAC10 Q969S8 6/20 0.65
HDAC11 Q96DB2 6/20 0.65
HDAC8 Q9BY41 6/20 0.65
HDAC6 Q9UBN7 6/20 0.65
HDAC9 Q9UKV0 6/20 0.65
HDAC5 Q9UQL6 6/20 0.65
PDGFRB P09619 3/20 0.62
GSK3B P49841 2/20 0.62
ARAF P10398 2/20 0.62
BRAF P15056 2/20 0.62
MEN1 O00255 1/20 0.62
PLK4 O00444 1/20 0.62
CIT O14578 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL940018 0.93 RAF1 (1.00) RAF1KDRHDAC3HDAC4HDAC1
SCHEMBL2480623 0.89 RAF1 (0.84) RAF1KDRHDAC3HDAC4HDAC1
SCHEMBL549001 0.89 RAF1 (1.00) RAF1KDRHDAC3HDAC4HDAC1
SCHEMBL548328 0.86 RAF1 (0.79) RAF1KDRHDAC3HDAC4HDAC1
SCHEMBL13471762 0.83 RAF1 (0.84) RAF1KDRHDAC3HDAC4HDAC1
SCHEMBL937568 0.82 RAF1 (1.00) RAF1KDRHDAC3HDAC4HDAC1
SCHEMBL3707691 0.82 RAF1 (0.83) RAF1KDRHDAC3HDAC4HDAC1
SCHEMBL2507080 0.82 RAF1 (0.75) RAF1KDRHDAC3HDAC4HDAC1
SCHEMBL3181311 0.81 RAF1 (0.70) RAF1KDRPDGFRBGSK3BARAF
SCHEMBL13471761 0.81 RAF1 (0.84) RAF1KDRHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1580188-B9 Aryl ureas as kinase inhibitors BAYER HEALTHCARE LLC (US) 2012-05-23 EP claimed
EP-1580188-B1 Aryl ureas as kinase inhibitors BAYER HEALTHCARE LLC (US) 2011-10-19 EP claimed