SCHEMBL24784175

SCHEMBL24784175

COc1ccc(-c2noc(-c3ccc(NCCN4CCN(C)CC4)nn3)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CXCR1 P25024 2/20 0.48
NPC1 O15118 5/20 0.44
RAB9A P51151 5/20 0.44
ACHE P22303 1/20 0.43
MAPT P10636 6/20 0.42
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NPSR1 Q6W5P4 1/20 0.42
S1PR1 P21453 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
TSHR P16473 2/20 0.42
LMNA P02545 1/20 0.42
STAT3 P40763 1/20 0.41
GAA P10253 1/20 0.41
TP53 P04637 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24783593 0.94 CXCR1 (0.51) CXCR1NPC1RAB9AACHEMAPT
SCHEMBL30133015 0.94 CXCR1 (0.51) CXCR1NPC1RAB9AACHEMAPT
SCHEMBL24784177 0.93 ACHE (0.51) NPC1RAB9AACHEMAPTPOLB
SCHEMBL24784178 0.91 NPC1 (0.56) NPC1RAB9AMAPTNPSR1TSHR
SCHEMBL30133010 0.91 NPC1 (0.56) NPC1RAB9AMAPTNPSR1TSHR
SCHEMBL30133020 0.87 ACP1 (0.48) CXCR1NPC1RAB9AACHEMAPT
SCHEMBL24783591 0.87 ACP1 (0.48) CXCR1NPC1RAB9AACHEMAPT
SCHEMBL24783691 0.87 ACP1 (0.49) CXCR1ACHEMAPTPOLBSMN1; SMN2
SCHEMBL24784179 0.84 TSHR (0.57) CXCR1MAPTPOLBSMN1; SMN2TSHR
SCHEMBL30133014 0.84 TSHR (0.57) CXCR1MAPTPOLBSMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022261296-A1 COMPOUNDS THAT BIND NON-CANONICAL G-QUADRUPLEX STRUCTURES AND METHODS OF MAKING AND USING THE SAME THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2022-12-15 WO disclosed