SCHEMBL2478684

SCHEMBL2478684

O=C(O)N1CCN(c2c(F)cc(N3C[C@H](Cn4cc(CF)nn4)OC3=O)cc2F)CC1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOA P21397 16/20 0.49
KCNH2 Q12809 2/20 0.44
MAOB P27338 3/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18059592 0.88 MAOA (0.49) MAOAKCNH2MAOB
SCHEMBL2501174 0.88 MAOA (0.49) MAOAKCNH2MAOB
SCHEMBL2478686 0.81 MAOA (0.33) MAOA
SCHEMBL2509465 0.81 MAOA (0.50) MAOAKCNH2MAOB
SCHEMBL18059602 0.81 MAOA (0.50) MAOAKCNH2MAOB
SCHEMBL12197576 0.80 MAOA (0.41) MAOAKCNH2
SCHEMBL18059599 0.80 CYP3A4 (0.42) MAOAKCNH2CYP3A4CYP2D6
SCHEMBL12196635 0.80 CYP3A4 (0.42) MAOAKCNH2CYP3A4CYP2D6
SCHEMBL12197566 0.79 MAOA (0.40) MAOAKCNH2MAOBCYP3A4CYP2D6
SCHEMBL4488687 0.78 MAOA (0.57) MAOAKCNH2MAOBCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367820-A2 Novel antimicrobials Panacea Biotec Limited (IN) 2011-09-28 EP disclosed
WO-2010058423-A2 NOVEL ANTIMICROBIALS PANACEA BIOTEC LTD. (IN) 2010-05-27 WO disclosed