SCHEMBL24802124

SCHEMBL24802124

CNCCNC1CN(C(C)=O)C1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.40
CHRNA3 P32297 3/20 0.40
CHRNA4 P43681 3/20 0.40
CHRNB4 P30926 2/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNB3 Q05901 1/20 0.39
CHRNA6 Q15825 1/20 0.39
EPHX2 P34913 6/20 0.36
EPHX1 P07099 2/20 0.36
OPRL1 P41146 1/20 0.35
CARM1 Q86X55 3/20 0.35
PRMT6 Q96LA8 3/20 0.35
CYP1A2 P05177 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PRMT8 Q9NR22 2/20 0.33
KISS1R Q969F8 1/20 0.33
PRMT1 Q99873 1/20 0.33
PIK3CD O00329 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21600937 0.84 CHRNB2 (0.42) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA7
SCHEMBL20030841 0.79 GAA (0.40) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA7
SCHEMBL17572858 0.78 CHRNB2 (0.44) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA7
SCHEMBL24207985 0.78 CHRNB2 (0.33) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA7
SCHEMBL2102558 0.76 CHRNB2 (0.42) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA7
SCHEMBL3832771 0.74
SCHEMBL8151297 0.73 OPRL1 (0.46) EPHX2EPHX1OPRL1
SCHEMBL8138756 0.73 OPRL1 (0.46) EPHX2EPHX1OPRL1
SCHEMBL25026706 0.73 CARM1 (0.39) CARM1PRMT6PRMT8PRMT1
SCHEMBL24481225 0.72 EPHX2 (0.50) EPHX2EPHX1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022268052-A9 (R) -GLUTARIMIDE CRBN LIGANDS AND METHODS OF USE BEIGENE, LTD. (KY) 2023-08-17 WO disclosed
WO-2022268052-A1 (R) -GLUTARIMIDE CRBN LIGANDS AND METHODS OF USE BEIGENE, LTD. (KY) 2022-12-29 WO disclosed