SCHEMBL24822802

SCHEMBL24822802

COc1c(-c2cnn(C)n2)ccc(F)c1N

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 9/20 0.35
FEN1 P39748 9/20 0.35
TYK2 P29597 5/20 0.34
AOC3 Q16853 2/20 0.33
AR P10275 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM3 P20309 1/20 0.31
BRD4 O60885 1/20 0.30
BRD3 Q15059 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20150274 0.85 TYK2 (0.33) ALOX5APFEN1TYK2AOC3CHRM2
SCHEMBL24775869 0.77 AOC3 (0.33) ALOX5APFEN1TYK2AOC3CHRM2
SCHEMBL30079490 0.77 TYK2 (0.41) TYK2AOC3CHRM2CHRM3
SCHEMBL15698663 0.77 TYK2 (0.41) TYK2AOC3CHRM2CHRM3
SCHEMBL30079457 0.75 TYK2 (0.35) ALOX5APFEN1TYK2AOC3CHRM2
SCHEMBL24776721 0.75 TYK2 (0.35) ALOX5APFEN1TYK2AOC3CHRM2
SCHEMBL24822834 0.75 TYK2 (0.35) ALOX5APFEN1TYK2AOC3CHRM2
SCHEMBL29947295 0.75 TYK2 (0.35) ALOX5APFEN1TYK2AOC3CHRM2
SCHEMBL24776105 0.74 FYN (0.33) ALOX5APFEN1TYK2AOC3CHRM2
SCHEMBL29947259 0.74 FYN (0.33) ALOX5APFEN1TYK2AOC3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250163004-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY 2025-05-22 US disclosed
US-20240190829-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY 2024-06-13 US disclosed
CN-117794912-A Substituted heterocyclic compounds 百时美施贵宝公司 2024-03-29 CN disclosed
EP-4337655-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS Bristol-Myers Squibb Company (US) 2024-03-20 EP disclosed
US-11866414-B2 Substituted heterocyclic compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2024-01-09 US disclosed
US-20220411384-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY 2022-12-29 US disclosed
US-20220411384-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY 2022-12-29 US disclosed
WO-2022241171-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2022-11-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11866414-B2 Substituted heterocyclic compounds TYK2, JAK2, STAT3 ALOX5AP 3808/4885FEN1 4033/4885TYK2 1/4885
US-20250163004-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS TYK2, JAK2, STAT3 ALOX5AP 3808/4885FEN1 4033/4885TYK2 1/4885
US-20220411384-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS TYK2, JAK2, STAT3 ALOX5AP 3808/4885FEN1 4033/4885TYK2 1/4885
US-20240190829-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS TYK2, JAK2, STAT3 ALOX5AP 3808/4885FEN1 4033/4885TYK2 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.