SCHEMBL24823375

SCHEMBL24823375

Cc1cc2cc3c(cc2nc1C(C)(C)O)C(=O)NC3

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.39
PIM1 P11309 6/20 0.36
CLK4 Q9HAZ1 3/20 0.36
GSK3B P49841 3/20 0.36
NTRK1 P04629 2/20 0.36
FLT3 P36888 2/20 0.36
DAPK3 O43293 1/20 0.36
ROCK1 Q13464 1/20 0.36
PIM2 Q9P1W9 5/20 0.35
PIM3 Q86V86 2/20 0.35
DYRK1B Q9Y463 2/20 0.35
FYN P06241 1/20 0.35
MKNK2 Q9HBH9 4/20 0.33
MKNK1 Q9BUB5 3/20 0.33
MAPK1 P28482 1/20 0.33
F9 P00740 1/20 0.32
NTRK2 Q16620 2/20 0.32
TYRO3 Q06418 1/20 0.32
TBK1 Q9UHD2 1/20 0.32
JAK2 O60674 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24823391 0.86 CYP17A1 (0.38) CYP17A1PIM1CLK4GSK3BNTRK1
SCHEMBL30310922 0.86 CYP17A1 (0.38) CYP17A1PIM1CLK4GSK3BNTRK1
SCHEMBL29871724 0.68 CLK4 (0.49) CYP17A1PIM1CLK4GSK3BNTRK1
SCHEMBL10139776 0.68 HTT (0.52) PIM1CLK4GSK3BNTRK1FLT3
SCHEMBL31195434 0.68 HTT (0.52) PIM1CLK4GSK3BNTRK1FLT3
SCHEMBL5230177 0.67 PARP1 (0.46) PIM1CLK4GSK3BNTRK1FLT3
SCHEMBL29010946 0.67 NTRK2 (0.35) CYP17A1CLK4GSK3BNTRK1FLT3
SCHEMBL29010943 0.66 KDM4E (0.38) MAPK1
SCHEMBL30310966 0.66 KDM4E (0.38) MAPK1
SCHEMBL31741758 0.66 MKNK2 (0.51) CYP17A1CLK4GSK3BNTRK1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022267930-A1 TRICYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 中国医药研究开发中心有限公司 2022-12-29 WO disclosed