SCHEMBL2482903

SCHEMBL2482903

O=C(N[C@@H](CO)Cc1ccccc1)OCc1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 2/20 0.76
CYP3A4 P08684 6/20 0.57
MAPK1 P28482 1/20 0.57
ALDH1A1 P00352 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
TSHR P16473 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
TACR1 P25103 2/20 0.56
CTSL P07711 2/20 0.54
CTSK P43235 2/20 0.54
CTSB P07858 1/20 0.54
CTSS P25774 1/20 0.54
TRPM8 Q7Z2W7 1/20 0.53
ALOX15 P16050 1/20 0.53
BACE1 P56817 1/20 0.53
SYK P43405 1/20 0.52
ATM Q13315 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1051352 1.00 CTRB1 (0.76) CTRB1CYP3A4MAPK1ALDH1A1CYP1A2
SCHEMBL2435512 1.00 CTRB1 (0.76) CTRB1CYP3A4MAPK1ALDH1A1CYP1A2
Carbamic Acid SCHEMBL8426387 0.96 CTRB1 (0.70) CTRB1CYP3A4MAPK1ALDH1A1CYP1A2
Carbamic Acid SCHEMBL8426357 0.96 CTRB1 (0.70) CTRB1CYP3A4MAPK1ALDH1A1CYP1A2
SCHEMBL3126143 0.94 CTRB1 (0.68) CTRB1CYP3A4MAPK1ALDH1A1CYP1A2
SCHEMBL8612701 0.94 CTRB1 (0.68) CTRB1CYP3A4MAPK1ALDH1A1CYP1A2
SCHEMBL7342331 0.93 CTRB1 (0.67) CTRB1CYP3A4MAPK1ALDH1A1CYP1A2
SCHEMBL4829896 0.92 CTRB1 (0.68) CTRB1ALDH1A1CYP1A2SMN1; SMN2TACR1
SCHEMBL7301416 0.91 CTRB1 (0.64) CTRB1CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL9484576 0.91 CTRB1 (0.64) CTRB1CYP3A4CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4633581-A1 A TOPICAL COMPOSITION Rock & Herb Pte Ltd (SG) 2025-10-22 EP claimed
WO-2024128980-A1 A TOPICAL COMPOSITION ROCK & HERB PTE LTD (SG) 2024-06-20 WO claimed
EP-0815074-B1 O-CARBAMOYL-(D)-PHENYLALANILOL COMPOUNDS AND PROCESS FOR PREPARING THE SAME SK CORP (KR) 2001-10-04 EP claimed
EP-0728129-B1 NOVEL PHENYLALKYLAMINOALCOHOL CARBAMATES AND PROCESS FOR PREPARING THE SAME YUKONG LTD (KR) 1999-11-03 EP claimed
US-5955499-A PHARMACEUTICALS USEFUL TO TREAT DISEASES OF THE CENTRAL NERVOUS SYSTEM, I.E. ANTIDEPRESSANTS YUKONG LIMITED (KR) 1999-09-21 US claimed
EP-0815074-A1 O-CARBAMOYL-(D)-PHENYLALANILOL COMPOUNDS AND PROCESS FOR PREPARING THE SAME YUKONG LIMITED (KR) 1998-01-07 EP claimed
EP-0728129-A1 NOVEL PHENYLALKYLAMINOALCOHOL CARBAMATES AND PROCESS FOR PREPARING THE SAME YUKONG LIMITED (KR) 1996-08-28 EP claimed
WO-1996024577-A1 O-CARBAMOYL-(D)-PHENYLALANILOL COMPOUNDS AND PROCESS FOR PREPARING THE SAME YUKONG LIMITED (KR) 1996-08-15 WO claimed
WO-1996007637-A1 NOVEL PHENYLALKYLAMINOALCOHOL CARBAMATES AND PROCESS FOR PREPARING THE SAME YUKONG LIMITED (KR) 1996-03-14 WO claimed
EP-4688731-A1 PROCESS FOR PREPARING (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE INKE, S.A. (ES) 2026-02-11 EP disclosed
EP-4633581-A1 A TOPICAL COMPOSITION Rock & Herb Pte Ltd (SG) 2025-10-22 EP disclosed
WO-2024208791-A1 PROCESS FOR PREPARING (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE INKE, S.A. (ES) 2024-10-10 WO disclosed
US-20240208992-A1 MACROCYCLES AS CFTR MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2024-06-27 US disclosed
WO-2024128980-A1 A TOPICAL COMPOSITION ROCK & HERB PTE LTD (SG) 2024-06-20 WO disclosed
US-5157143-A DIASTEREOSELECTIVE PROCESS FOR THE PREPARATION OF INTERMEDIATES USEFUL FOR THE SYNTHESIS OF PEPTIDE DERIVATIVES ZAMBON GROUP S.P.A. (IT) 1992-10-20 US disclosed
EP-0341462-B1 DIASTEREOSELECTIVE PROCESS FOR THE PREPARATION OF INTERMEDIATES USEFUL FOR THE SYNTHESIS OF PEPTIDE DERIVATIVES ZAMBON GROUP S.p.A. (IT) 1992-09-09 EP disclosed
EP-0439556-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
WO-1990004917-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1990-05-17 WO disclosed
EP-0365992-A1 Heterocyclic peptide renin inhibitors ABBOTT LABORATORIES (US) 1990-05-02 EP disclosed
EP-0341462-A1 Diastereoselective process for the preparation of intermediates useful for the synthesis of peptide derivatives ZAMBON GROUP S.p.A. (IT) 1989-11-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240208992-A1 MACROCYCLES AS CFTR MODULATORS CFTR, PKD1, ARRB1 CTRB1 316/4885CYP3A4 1162/4885MAPK1 2666/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.