SCHEMBL2483716

SCHEMBL2483716

O=C(Nc1cccc(Oc2ccccc2)c1)N1CCc2c(c(Br)nc3[nH]ncc23)C1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 1/20 0.47
PDGFRB P09619 1/20 0.47
GOT1 P17174 1/20 0.45
TRPV1 Q8NER1 3/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
FAAH O00519 6/20 0.43
GPR142 Q7Z601 1/20 0.43
FLT3 P36888 1/20 0.41
S1PR2 O95136 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2486666 0.89 NPC1 (0.47) PDGFRBTRPV1NPC1RAB9AMAPT
SCHEMBL2483986 0.87 NPC1 (0.40) BRS3PDGFRBTRPV1NPC1RAB9A
SCHEMBL2806247 0.84 PDGFRB (0.52) BRS3PDGFRBGOT1NPC1RAB9A
SCHEMBL2805744 0.80 PDGFRB (0.48) BRS3PDGFRBGOT1NPC1RAB9A
SCHEMBL2490058 0.78 MAPT (0.44) TRPV1NPC1RAB9AALDH1A1MAPT
SCHEMBL2804674 0.77 BRS3 (0.50) BRS3PDGFRBGOT1TRPV1NPC1
SCHEMBL2802809 0.75 PDGFRB (0.62) PDGFRBTRPV1NPC1RAB9AFAAH
SCHEMBL2802299 0.74 NPC1 (0.61) NPC1RAB9AALDH1A1MAPTMAPK1
SCHEMBL2488481 0.74 ROCK2 (0.36) TRPV1ALDH1A1
SCHEMBL1000524 0.73 TRPV1 (0.73) TRPV1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379551-A1 SUBSTITUTED PYRAZOLO [3, 4-B]PYRIDINE COMPOUNDS ArQule, Inc. (US) 2011-10-26 EP disclosed
WO-2010078427-A1 SUBSTITUTED PYRAZOLO [3, 4-B] PYRIDINE COMPOUNDS ARQULE, INC. (US) 2010-07-08 WO disclosed