SCHEMBL2484253

SCHEMBL2484253

Cc1noc(-c2ccccc2)c1CN1CC2(CC1=O)C(=O)N(C(C(=O)O)C(C)(C)C)c1ccc(Cl)cc12

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 18/20 0.72
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2486050 0.90 PTGDR2 (0.74) PTGDR2HCRTR1HCRTR2
SCHEMBL2483121 0.84 PTGDR2 (0.65) PTGDR2
SCHEMBL2482558 0.84 PTGDR2 (1.00) PTGDR2
SCHEMBL11959127 0.83 PTGDR2 (0.82) PTGDR2
SCHEMBL2486047 0.82 PTGDR2 (0.95) PTGDR2
SCHEMBL2486611 0.80 PTGDR2 (0.59) PTGDR2
SCHEMBL2481296 0.79 PTGDR2 (0.66) PTGDR2
SCHEMBL2484605 0.73 PTGDR2 (0.72) PTGDR2HCRTR1HCRTR2
SCHEMBL2483157 0.70 PTGDR2 (1.00) PTGDR2
SCHEMBL2483198 0.68 PTGDR2 (0.38) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891075-B1 TRICYCLIC SPIRO DERIVATIVES AS CRTH2 MODULATORS MERCK SERONO SA (CH) 2011-10-19 EP disclosed