SCHEMBL2484828

SCHEMBL2484828

CN1[C@@H]2CC[C@H]1C[C@@H](Oc1ccc(-c3ccc4[nH]ccc4c3)nc1)C2

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 10/20 0.49
KCNH2 Q12809 6/20 0.49
CHRNB2 P17787 2/20 0.46
CHRNB4 P30926 2/20 0.46
CHRNA3 P32297 2/20 0.46
CHRNA4 P43681 2/20 0.46
CHRNA10 Q9GZZ6 1/20 0.46
CHRNA9 Q9UGM1 1/20 0.46
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
PDE10A Q9Y233 1/20 0.41
ABL1 P00519 1/20 0.40
LRRK2 Q5S007 1/20 0.39
FYN P06241 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2484827 1.00 CHRNA7 (0.49) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL744341 1.00 CHRNA7 (0.49) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL746332 0.92 CHRNA7 (0.48) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL746978 0.91 CHRNA7 (0.47) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL744535 0.88 CHRNA7 (0.41) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL746345 0.87 PRKCZ (0.43) SLC6A2SLC6A3
SCHEMBL744687 0.86 CHRNA7 (0.49) CHRNA7KCNH2SLC6A2SLC6A3
SCHEMBL743968 0.86 CHRNA7 (0.53) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL2481429 0.85 CHRNA7 (0.52) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL748372 0.84 KCNH2 (0.53) CHRNA7KCNH2SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2018380-B1 Cns active fused bicycloheterocycle substituted azabicyclic alkane derivatives ABBOTT LAB (US) 2011-10-19 EP claimed