SCHEMBL2485876

SCHEMBL2485876

COCc1cc(-c2nc(-c3ccc4c(c3)CN(CCC(=O)O)CC4)no2)ccc1-c1ccccc1C.COCc1cc(-c2nc(-c3ccc4c(c3)CN(CCC(=O)OC(C)(C)C)CC4)no2)ccc1-c1ccccc1C

nearest known ligand 0.88

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.88
S1PR3 Q99500 7/20 0.54
S1PR5 Q9H228 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2420128 0.97 S1PR1 (0.83) S1PR1S1PR3S1PR5
SCHEMBL2488515 0.94 S1PR1 (0.77) S1PR1S1PR3S1PR5
SCHEMBL2418025 0.94 S1PR1 (1.00) S1PR1S1PR3S1PR5
SCHEMBL2413218 0.91 S1PR1 (0.72) S1PR1S1PR3S1PR5
SCHEMBL2417129 0.91 S1PR1 (1.00) S1PR1S1PR3S1PR5
SCHEMBL2484873 0.89 S1PR1 (0.88) S1PR1S1PR3S1PR5
SCHEMBL2418804 0.87 S1PR1 (0.87) S1PR1S1PR3S1PR5
SCHEMBL2415296 0.87 S1PR1 (1.00) S1PR1S1PR3
SCHEMBL2416941 0.86 S1PR1 (0.82) S1PR1S1PR3S1PR5
SCHEMBL2417428 0.82 S1PR1 (1.00) S1PR1S1PR3S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376484-A1 OXADIAZOLE FUSED HETEROCYCLIC DERIVATIVES USEFUL FOR THE TREATMENT OF MULTIPLE SCLEROSIS Merck Serono S.A. (CH) 2011-10-19 EP disclosed
WO-2010069949-A1 OXADIAZOLE FUSED HETEROCYCLIC DERIVATIVES USEFUL FOR THE TREATMENT OF MULTIPLE SCLEROSIS MERCK SERONO S.A. (CH) 2010-06-24 WO disclosed