SCHEMBL24854597

SCHEMBL24854597

OB(O)c1c(F)ccc2c1cnn2C1CCCCO1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 5/20 0.44
CYP4A11 Q02928 5/20 0.44
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43
LMNA P02545 2/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
ATR Q13535 5/20 0.32
ESR1 P03372 1/20 0.32
MAPT P10636 1/20 0.32
PDE1A P54750 1/20 0.30
PDE1B Q01064 1/20 0.30
PDE1C Q14123 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21243927 0.86 RXRA (0.43) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL18128583 0.86 CYP4F2 (0.44) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL21243954 0.85 RXRA (0.41) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL21196043 0.84 CYP4F2 (0.49) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL28578639 0.84 CYP4F2 (0.43) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL31437298 0.84 RXRA (0.42) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL21196032 0.81 CYP4F2 (0.44) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL29478977 0.81 CYP4F2 (0.44) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL30959446 0.81 RXRA (0.40) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL23272983 0.81 CYP4F2 (0.44) CYP4F2CYP4A11RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250304537-A1 HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME REPARE THERAPEUTICS INC. (CA) 2025-10-02 US disclosed
CN-119894872-A Heteroarenes, pharmaceutical compositions containing heteroarenes, and methods of use thereof 修复治疗公司 2025-04-25 CN disclosed
EP-4526293-A1 HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME Repare Therapeutics Inc. (CA) 2025-03-26 EP disclosed
WO-2023220831-A1 HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME REPARE THERAPEUTICS INC. (CA) 2023-11-23 WO disclosed
US-11760744-B2 Fused ring compounds GENENTECH, INC. (US) 2023-09-19 US disclosed
US-11760744-B2 Fused ring compounds GENENTECH, INC. (US) 2023-09-19 US disclosed
US-20230002345-A1 FUSED RING COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2023-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250304537-A1 HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME CSNK1A1, CSNK1G1, CSNK2A1 CYP4F2 2157/4885CYP4A11 2492/4885RXRA 4196/4885
US-11760744-B2 Fused ring compounds KRAS, NRAS, HRAS CYP4F2 813/4885CYP4A11 1657/4885RXRA 1930/4885
US-20230002345-A1 FUSED RING COMPOUNDS KRAS, NRAS, HRAS CYP4F2 813/4885CYP4A11 1657/4885RXRA 1930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.