SCHEMBL24856005

SCHEMBL24856005

CCCN1CCC(c2ccccc2)(N(C)C(C)=O)CC1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 8/20 0.61
OPRL1 P41146 6/20 0.61
TACR3 P29371 3/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
TACR2 P21452 1/20 0.50
TACR1 P25103 1/20 0.50
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24855511 0.92 OPRM1 (0.52) OPRM1OPRL1TACR3CYP3A4CYP2D6
SCHEMBL24230841 0.88 OPRM1 (0.46) OPRM1OPRL1TACR3CYP3A4CYP2D6
SCHEMBL9910972 0.84 OPRM1 (0.71) OPRM1OPRL1TACR3CYP3A4CYP2D6
SCHEMBL4630038 0.83 OPRM1 (0.61) OPRM1OPRL1TACR3CYP3A4CYP2D6
SCHEMBL24855392 0.81 TACR3 (0.49) OPRM1OPRL1TACR3CYP3A4CYP2D6
SCHEMBL3410403 0.77 OPRM1 (1.00) OPRM1OPRL1
SCHEMBL3742048 0.76 TACR3 (0.62) OPRM1OPRL1TACR3
SCHEMBL3751174 0.76 TACR3 (0.62) OPRM1OPRL1TACR3
SCHEMBL6022898 0.75 OPRM1 (0.51) OPRM1OPRL1TACR3CYP3A4CYP2D6
SCHEMBL2333169 0.75 HRH3 (0.54) OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023147134-A2 METHODS FOR TREATING PATIENTS HAVING LOW ESTROGEN WITH NK3 ANTAGONISTS ACER THERAPEUTICS, INC. (US) 2023-08-03 WO disclosed
WO-2023147135-A1 NK RECEPTOR ANTAGONISTS FOR TREATMENT OF PROSTATE CANCER ACER THERAPEUTICS, INC. (US) 2023-08-03 WO disclosed
WO-2023278843-A2 SOLID FORMS OF OSANETANT ACER THERAPEUTICS, INC. (US) 2023-01-05 WO disclosed