SCHEMBL24865600

SCHEMBL24865600

CN1Cc2cc(Nc3ccc(N4CCC(C(F)(F)F)CC4)cc3)ccc2N(C)C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.45
BRD2 P25440 1/20 0.40
BRD3 Q15059 1/20 0.40
BCL6 P41182 1/20 0.34
CNR2 P34972 1/20 0.34
SYK P43405 2/20 0.33
DCLK1 O15075 1/20 0.33
LRRK2 Q5S007 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.32
EGFR P00533 2/20 0.32
JAK2 O60674 1/20 0.32
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
KCNH2 Q12809 1/20 0.32
NAMPT P43490 1/20 0.32
CDK4 P11802 2/20 0.32
CCND1 P24385 2/20 0.32
CCND2 P30279 2/20 0.32
CCND3 P30281 2/20 0.32
CTSC P53634 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31123328 1.00 BRD4 (0.45) BRD4BRD2BRD3BCL6CNR2
SCHEMBL24865338 0.84 TRIM24 (0.42) BRD4BCL6CNR2SYKEGFR
SCHEMBL24865619 0.83 BCL6 (0.36) BRD4BCL6CNR2SYKDCLK1
SCHEMBL24865514 0.83 KIT (0.44) BCL6CNR2SYK
SCHEMBL31123249 0.82 CNR2 (0.36) BRD4BCL6CNR2SYKDCLK1
SCHEMBL24865354 0.82 CNR2 (0.36) BRD4BCL6CNR2SYKDCLK1
SCHEMBL24865525 0.82 BCL6 (0.35) BCL6CNR2SYKDCLK1LRRK2
SCHEMBL24865651 0.81 DDB1 (0.44) BRD4BCL6CNR2DCLK1LRRK2
SCHEMBL31123277 0.80 CNR2 (0.36) BCL6CNR2SYKSCN10AEGFR
SCHEMBL24865078 0.79 KIT (0.33) BRD4BCL6CNR2EGFRJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed