SCHEMBL2487154

SCHEMBL2487154

CCOC(=O)C(Cl)=NNc1cccc(C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KYAT1 Q16773 1/20 0.52
GAA P10253 9/20 0.48
LMNA P02545 3/20 0.48
MAPT P10636 7/20 0.47
ALDH1A1 P00352 4/20 0.47
NPSR1 Q6W5P4 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
HPGD P15428 2/20 0.47
ATM Q13315 1/20 0.47
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
RECQL P46063 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ALOX12 P18054 1/20 0.45
TP53 P04637 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8060308 1.00 KYAT1 (0.52) KYAT1GAALMNAMAPTALDH1A1
SCHEMBL1998080 1.00 KYAT1 (0.52) KYAT1GAALMNAMAPTALDH1A1
SCHEMBL5252880 0.87 KYAT1 (0.67) KYAT1GAALMNAMAPTALDH1A1
SCHEMBL5252876 0.87 KYAT1 (0.67) KYAT1GAALMNAMAPTALDH1A1
SCHEMBL31597961 0.87 KYAT1 (0.67) KYAT1GAALMNAMAPTALDH1A1
SCHEMBL6107763 0.87 KYAT1 (0.67) KYAT1GAALMNAMAPTALDH1A1
SCHEMBL11762275 0.86 KYAT1 (0.50) KYAT1GAALMNAMAPTALDH1A1
SCHEMBL11762267 0.86 KYAT1 (0.50) KYAT1GAALMNAMAPTALDH1A1
SCHEMBL25985823 0.86 KYAT1 (0.50) KYAT1GAALMNAMAPTALDH1A1
SCHEMBL16730435 0.86 KYAT1 (0.50) KYAT1GAALMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379531-A1 PROCESSES FOR THE MANUFACTURE OF 3-{4-METHYL-5- [ (IR) -1- (2- (3-METHYLPHENYL) -2H-TETRAZOL-5-YL) -ETHOXY]-4H- [1,2, 4]TRIAZOL-3-YL} -PYRIDINE, 4-METHYL-3-METHYLTHIO-5- (3- PYRIDYL)-L,2,4-TRIAZOLE, AND (IR) -1- [2- (3-METHYLPHENYL) -2H- TETRAZOL-5-YL]ETHANOL AstraZeneca AB (SE) 2011-10-26 EP disclosed