SCHEMBL2489034

SCHEMBL2489034

CC(C)(C)N1CCC[C@@H](Nc2ncc3c(n2)-c2ccccc2[C@H](c2ccc(Cl)c(Cl)c2)C3)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 5/20 0.41
CCNK O75909 4/20 0.41
CDK12 Q9NYV4 4/20 0.41
CCNT1 O60563 3/20 0.41
CDK9 P50750 3/20 0.41
CCNE1 P24864 2/20 0.41
CDK7 P50613 3/20 0.40
CCNH P51946 3/20 0.40
MNAT1 P51948 3/20 0.40
FGFR1 P11362 1/20 0.39
FGFR2 P21802 1/20 0.39
JUN P05412 4/20 0.38
MAPK8 P45983 4/20 0.38
MAPK9 P45984 4/20 0.38
MAPK10 P53779 3/20 0.38
ADORA1 P30542 1/20 0.37
SLC6A2 P23975 5/20 0.36
SLC6A4 P31645 5/20 0.36
SLC6A3 Q01959 5/20 0.36
CYP2D6 P10635 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2493170 0.87 MAPK1 (0.45) CDK2CCNKCDK12CCNT1CDK9
SCHEMBL2493168 0.87 MAPK1 (0.45) CDK2CCNKCDK12CCNT1CDK9
SCHEMBL2492524 0.87 MAPK1 (0.45) CDK2CCNKCDK12CCNT1CDK9
SCHEMBL2492527 0.87 MAPK1 (0.45) CDK2CCNKCDK12CCNT1CDK9
SCHEMBL2492528 0.87 MAPK1 (0.45) CDK2CCNKCDK12CCNT1CDK9
SCHEMBL16360384 0.85 MAPK10 (0.44) CDK2CCNKCDK12CCNT1CDK9
SCHEMBL16360406 0.85 MAPK10 (0.44) CDK2CCNKCDK12CCNT1CDK9
SCHEMBL2488139 0.82 MAPK8 (0.46) CDK2CCNT1JUNMAPK8MAPK9
SCHEMBL13126036 0.81 MAPK3 (0.37) CCNKCDK12CCNT1CDK9CDK7
SCHEMBL2804817 0.80 FGFR1 (0.41) FGFR1FGFR2SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379506-A1 SUBSTITUTED 5,6-DIHYDRO-6-PHENYLBENZO[F]ISOQUINOLIN-2-AMINE COMPOUNDS ArQule, Inc. (US) 2011-10-26 EP disclosed
WO-2010078421-A1 SUBSTITUTED 5,6-DIHYDRO-6-PHENYLBENZO[F] ISOQUINOLIN-2-AMINE COMPOUNDS ARQULE, INC. (US) 2010-07-08 WO disclosed