SCHEMBL2489158

SCHEMBL2489158

Brc1cnc(-c2sc(Nc3ccccn3)nc2-c2ccccn2)cc1Oc1cccc2ncccc12

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 4/20 0.37
PDE10A Q9Y233 3/20 0.36
KDR P35968 2/20 0.36
GRM4 Q14833 2/20 0.36
BRAF P15056 1/20 0.35
MECP2 P51608 1/20 0.35
KCNN1 Q92952 1/20 0.35
KCNN2 Q9H2S1 1/20 0.35
MBD2 Q9UBB5 1/20 0.35
KCNN3 Q9UGI6 1/20 0.35
KCNH2 Q12809 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33
GCK P35557 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
PTK2 Q05397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL190948 0.77 KCNN1 (0.49) MECP2KCNN1KCNN2MBD2KCNN3
SCHEMBL191010 0.71 NPC1 (0.48) GRM4KCNH2
SCHEMBL190731 0.70 GCK (0.45) BRAFGCK
SCHEMBL2493080 0.69 KCNN1 (0.42) TGFBR1KDRGRM4MECP2KCNN1
SCHEMBL6372588 0.68 MECP2 (0.55) KDRGRM4MECP2KCNN1KCNN2
SCHEMBL191400 0.67 GCK (0.44) BRAFGCK
Bromide SCHEMBL5174776 0.67 MECP2 (0.54) KDRGRM4MECP2KCNN1KCNN2
SCHEMBL5171103 0.65 MECP2 (0.51) KDRGRM4MECP2KCNN1KCNN2
SCHEMBL191875 0.64 NPC1 (0.43) TGFBR1PDE10AKDRBRAF
SCHEMBL191705 0.63 GCK (0.37) BRAFGCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8022222-B2 Glucokinase activators ARRAY BIOPHARMA, INC. (US) 2011-09-20 US disclosed