SCHEMBL24891764

SCHEMBL24891764

COC(=O)c1ccc(C(=O)Nc2ccc(CNC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.65
HDAC1 Q13547 3/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
ATM Q13315 1/20 0.53
MAPT P10636 3/20 0.53
TDP1 Q9NUW8 2/20 0.53
HDAC6 Q9UBN7 1/20 0.53
LMNA P02545 2/20 0.52
HPGD P15428 1/20 0.52
PTPN1 P18031 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
EPHX2 P34913 1/20 0.50
NR1H4 Q96RI1 1/20 0.50
MAPK1 P28482 1/20 0.50
PSMD14 O00487 1/20 0.50
CACNA1B Q00975 1/20 0.50
APBA1 Q02410 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23899245 0.94 NAMPT (0.72) NAMPTHDAC1MAPTTDP1HDAC6
SCHEMBL23899122 0.91 NAMPT (0.66) NAMPTHDAC1MAPTTDP1HDAC6
SCHEMBL26032300 0.90 MEN1 (0.57) NAMPTHDAC1CA1CA2NPC1
SCHEMBL1206337 0.89 NAMPT (0.55) NAMPTHDAC1CA1CA2NPC1
SCHEMBL24891652 0.89 NAMPT (0.66) NAMPTHDAC1MAPTTDP1HDAC6
SCHEMBL2213535 0.88 NAMPT (0.65) NAMPTHDAC1NPC1RAB9AMAPT
SCHEMBL24891860 0.88 NAMPT (0.65) NAMPTHDAC1MAPTTDP1HDAC6
SCHEMBL24670224 0.88 NAMPT (0.65) NAMPTHDAC1MAPTTDP1HDAC6
SCHEMBL24891767 0.86 NAMPT (0.58) NAMPTHDAC1MAPTTDP1HDAC6
SCHEMBL24891782 0.86 NAMPT (0.55) NAMPTHDAC1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed