SCHEMBL24891782

SCHEMBL24891782

COC(=O)c1ccc(C(=O)Nc2ccc(CNC(=O)OC(C)(C)C)cc2)cc1C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 5/20 0.55
SMN1; SMN2 Q16637 2/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
HDAC1 Q13547 3/20 0.49
HDAC6 Q9UBN7 1/20 0.48
TDP1 Q9NUW8 4/20 0.48
MAPT P10636 4/20 0.48
NPSR1 Q6W5P4 2/20 0.45
XBP1 P17861 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45
ROCK2 O75116 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
NR1H4 Q96RI1 2/20 0.44
LCK P06239 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
EPHX2 P34913 1/20 0.42
LMNA P02545 1/20 0.42
FPR3 P25089 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30182354 1.00 NAMPT (0.55) NAMPTSMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL30182158 0.92 NAMPT (0.58) NAMPTSMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL24891917 0.92 NAMPT (0.58) NAMPTSMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL30182509 0.90 NAMPT (0.56) NAMPTSMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL24891974 0.90 NAMPT (0.56) NAMPTSMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL24891759 0.87 NAMPT (0.53) NAMPTSMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL30182363 0.87 NAMPT (0.53) NAMPTSMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL24891764 0.86 NAMPT (0.65) NAMPTSMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL23898926 0.85 NAMPT (0.57) NAMPTSMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL30964980 0.85 NR1H4 (0.48) NAMPTSMN1; SMN2HDAC1NR1H4L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed