SCHEMBL24891773

SCHEMBL24891773

COc1cc(C2=CCN(C(=O)OC(C)(C)C)CC2)ccc1NC(=O)c1ccc(C(=O)Nc2ccc(CNC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.48
HDAC1 Q13547 3/20 0.46
KIT P10721 2/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
WNT3A P56704 1/20 0.42
MEN1 O00255 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
GRM5 P41594 1/20 0.41
GRM1 Q13255 1/20 0.41
CFTR P13569 2/20 0.40
QDPR P09417 1/20 0.40
CDK7 P50613 1/20 0.40
CDK13 Q14004 1/20 0.40
CDK12 Q9NYV4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24891779 0.91 HDAC1 (0.47) NAMPTHDAC1MAPTHDAC6ALDH1A1
SCHEMBL24670226 0.91 NAMPT (0.57) NAMPTHDAC1KITSMN1; SMN2MAPT
SCHEMBL24892276 0.91 NAMPT (0.57) NAMPTHDAC1KITSMN1; SMN2MAPT
SCHEMBL24891842 0.88 NAMPT (0.45) NAMPTHDAC1KITSMN1; SMN2MAPT
SCHEMBL24891939 0.85 NAMPT (0.38) NAMPTHDAC1MAPTHDAC6ALDH1A1
SCHEMBL24892051 0.84 NAMPT (0.53) NAMPTHDAC1KITSMN1; SMN2MAPT
SCHEMBL30182051 0.84 NAMPT (0.53) NAMPTHDAC1KITSMN1; SMN2MAPT
SCHEMBL30182548 0.84 NAMPT (0.54) NAMPTHDAC1KITSMN1; SMN2MAPT
SCHEMBL24891686 0.84 NAMPT (0.50) NAMPTHDAC1KITSMN1; SMN2MAPT
SCHEMBL24892325 0.84 NAMPT (0.50) NAMPTHDAC1KITSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed