SCHEMBL24897632

SCHEMBL24897632

C=C(C)CC(C)(N)COc1ccc(-c2ccnc(NC(C)=O)c2)nc1C(F)F

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 20/20 0.67
BMP2K Q9NSY1 4/20 0.67
GAK O14976 3/20 0.67
DAPK1 P53355 3/20 0.67
MKNK2 Q9HBH9 3/20 0.67
DAPK3 O43293 2/20 0.67
JAK2 O60674 2/20 0.67
HIPK4 Q8NE63 2/20 0.67
ROCK2 O75116 1/20 0.67
TYRO3 Q06418 1/20 0.67
DMPK Q09013 1/20 0.67
MKNK1 Q9BUB5 3/20 0.54
CIT O14578 2/20 0.54
KCNH2 Q12809 2/20 0.54
SLC6A2 P23975 1/20 0.54
LATS2 Q9NRM7 1/20 0.54
ABCG2 Q9UNQ0 1/20 0.54
CYP3A4 P08684 2/20 0.54
MYLK2 Q9H1R3 2/20 0.51
MAP2K1 Q02750 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24897651 1.00 AAK1 (0.67) AAK1BMP2KGAKDAPK1MKNK2
SCHEMBL27220561 0.94 AAK1 (0.66) AAK1BMP2KGAKDAPK1MKNK2
SCHEMBL27220555 0.94 AAK1 (0.66) AAK1BMP2KGAKDAPK1MKNK2
SCHEMBL24897655 0.93 AAK1 (0.78) AAK1BMP2KGAKDAPK1MKNK2
SCHEMBL24897623 0.93 AAK1 (0.78) AAK1BMP2KGAKDAPK1MKNK2
SCHEMBL24897683 0.88 AAK1 (0.68) AAK1BMP2KGAKDAPK1MKNK2
SCHEMBL24897634 0.88 AAK1 (0.68) AAK1BMP2KGAKDAPK1MKNK2
SCHEMBL24897796 0.85 AAK1 (0.73) AAK1BMP2KGAKDAPK1MKNK2
SCHEMBL24897596 0.85 AAK1 (0.73) AAK1BMP2KGAKDAPK1MKNK2
SCHEMBL24897659 0.85 AAK1 (0.73) AAK1BMP2KGAKDAPK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117715899-A AAK1 inhibitors and uses thereof 西藏海思科制药有限公司 2024-03-15 CN disclosed
WO-2023284838-A1 AAK1 INHIBITOR AND USE THEREOF 四川海思科制药有限公司 2023-01-19 WO disclosed