SCHEMBL24902207

SCHEMBL24902207

CC(C)Cc1ccc([C@H](C)C(=O)OCn2ccc3c(-c4cnn([C@@H](C)CC#N)c4)ncnc32)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
PTGS1 P23219 1/20 0.37
SLC6A2 P23975 1/20 0.37
JAK2 O60674 7/20 0.35
JAK1 P23458 6/20 0.35
JAK3 P52333 4/20 0.35
TYK2 P29597 3/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
TPH1 P17752 1/20 0.35
PTGS2 P35354 6/20 0.34
DAPK3 O43293 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24902082 0.89 JAK2 (0.49) JAK2JAK1JAK3TYK2HDAC6
SCHEMBL30864342 0.89 JAK2 (0.49) JAK2JAK1JAK3TYK2HDAC6
SCHEMBL24902070 0.89 JAK2 (0.49) JAK2JAK1JAK3TYK2HDAC6
SCHEMBL24902208 0.86 KDM5A (0.36) PGRADORA3PTGS1SLC6A2JAK2
SCHEMBL24902012 0.84 PTGS1 (0.39) PGRPTGS1PTGS2
SCHEMBL26610797 0.82 JAK2 (0.49) JAK2JAK1JAK3TYK2HDAC6
SCHEMBL24902066 0.81 PTGS1 (0.40) PGRADORA3PTGS1SLC6A2TPH1
SCHEMBL24902014 0.80 JAK1 (0.52) JAK2JAK1JAK3TYK2RET
SCHEMBL24902114 0.80 JAK1 (0.52) JAK2JAK1JAK3TYK2RET
SCHEMBL30223620 0.80 JAK1 (0.52) JAK2JAK1JAK3TYK2RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023001045-A9 EXTERNAL ANTI-INFLAMMATORY COUPLING COMPOUND DRUG, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海椿安生物医药科技有限公司 2023-10-26 WO disclosed
WO-2023001045-A1 EXTERNAL ANTI-INFLAMMATORY COUPLING COMPOUND DRUG, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海椿安生物医药科技有限公司 2023-01-26 WO disclosed