SCHEMBL2490533

SCHEMBL2490533

COc1c(C=Cc2ccccc2)cc(-c2ccn[nH]c2=O)cc1C(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.54
TNFRSF1A P19438 2/20 0.42
TUBB4A P04350 4/20 0.36
TUBB P07437 4/20 0.36
TUBA3C P0DPH7 4/20 0.36
TUBA1B P68363 4/20 0.36
TUBA4A P68366 4/20 0.36
TUBB4B P68371 4/20 0.36
TUBB3 Q13509 4/20 0.36
TUBB2A Q13885 4/20 0.36
TUBB8 Q3ZCM7 4/20 0.36
TUBA3E Q6PEY2 4/20 0.36
TUBA1A Q71U36 4/20 0.36
TUBA1C Q9BQE3 4/20 0.36
TUBB6 Q9BUF5 4/20 0.36
TUBB2B Q9BVA1 4/20 0.36
TUBB1 Q9H4B7 4/20 0.36
NFE2L2 Q16236 2/20 0.36
ERBB2 P04626 2/20 0.35
SNCA P37840 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2490531 1.00 CYP3A4 (0.54) CYP3A4TNFRSF1ATUBB4ATUBBTUBA3C
SCHEMBL6832451 0.90 CYP3A4 (0.52) CYP3A4TNFRSF1ATUBB4ATUBBTUBA3C
SCHEMBL2489645 0.85 CYP3A4 (0.73) CYP3A4TNFRSF1AERBB2SNCAFYN
SCHEMBL2489644 0.85 CYP3A4 (0.73) CYP3A4TNFRSF1AERBB2SNCAFYN
SCHEMBL1764331 0.83 CYP3A4 (0.74) CYP3A4TNFRSF1ATUBB4ATUBBTUBA3C
SCHEMBL1764330 0.83 CYP3A4 (0.74) CYP3A4TNFRSF1ATUBB4ATUBBTUBA3C
SCHEMBL6832515 0.82 CYP3A4 (0.43) CYP3A4PTGS2
SCHEMBL1764839 0.79 CYP3A4 (0.65) CYP3A4SNCAFYN
SCHEMBL6832471 0.79 PTGS2 (0.38) CYP3A4ERBB2EGFRADORA2AADORA1
SCHEMBL1542800 0.78 CYP3A4 (0.70) CYP3A4TNFRSF1ANFE2L2ERBB2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379534-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2011-10-26 EP claimed
WO-2010072598-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-07-01 WO claimed
US-20100158860-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS STEINER SANDRA 2010-06-24 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100158860-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS RFC1, RRP1B, RRBP1 CYP3A4 978/4885TNFRSF1A 3504/4885TUBB4A 1918/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.