SCHEMBL24906222

SCHEMBL24906222

CS(=O)(=O)c1cc(NC(=O)c2c(CC(F)(F)F)c(C3CC3)nn2CC2CCOCC2)ccn1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 13/20 0.42
RAF1 P04049 5/20 0.36
BRAF P15056 5/20 0.36
NR3C1 P04150 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30141432 1.00 SCN10A (0.42) SCN10ARAF1BRAFNR3C1AKR1C3
SCHEMBL24906422 0.89 SCN10A (0.44) SCN10ARAF1BRAFAKR1C3AKR1C2
SCHEMBL30141382 0.86 SCN10A (0.40) SCN10ARAF1BRAFNR3C1
SCHEMBL24906218 0.86 SCN10A (0.40) SCN10ARAF1BRAFNR3C1
SCHEMBL24758389 0.84 SCN10A (0.38) SCN10ARAF1BRAFNR3C1
SCHEMBL30141366 0.79 SCN10A (0.45) SCN10A
SCHEMBL24906328 0.79 SCN10A (0.45) SCN10A
SCHEMBL24906504 0.78 SCN10A (0.45) SCN10A
SCHEMBL24906303 0.77 SCN10A (0.43) SCN10A
SCHEMBL24906475 0.76 SCN10A (0.43) SCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230025025-A1 SUBSTITUTED PYRAZOLE AMIDES GRUENENTHAL GMBH (DE) 2023-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230025025-A1 SUBSTITUTED PYRAZOLE AMIDES SCN8A, SCN1A, SCN7A SCN10A 8/4885RAF1 934/4885BRAF 1456/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.