SCHEMBL24912178

SCHEMBL24912178

C=CC[C@@H](C)S(=O)(=O)N(Cc1ccc(O)cc1)Cc1ccc(OC)cc1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
APLNR P35414 16/20 0.54
TAS2R14 Q9NYV8 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24912180 1.00 APLNR (0.54) APLNRTAS2R14L3MBTL1
SCHEMBL17542305 0.94 APLNR (0.61) APLNRTAS2R14L3MBTL1
SCHEMBL17542070 0.94 APLNR (0.61) APLNRTAS2R14L3MBTL1
SCHEMBL17542467 0.94 APLNR (0.61) APLNRTAS2R14L3MBTL1
SCHEMBL20630302 0.88 APLNR (0.52) APLNRTAS2R14L3MBTL1
SCHEMBL24912187 0.86 APLNR (0.52) APLNRTAS2R14
SCHEMBL20670351 0.82 APLNR (0.46) APLNRTAS2R14
SCHEMBL23670695 0.81 APLNR (0.58) APLNRTAS2R14L3MBTL1
SCHEMBL19284930 0.81 APLNR (0.58) APLNRTAS2R14L3MBTL1
SCHEMBL23670755 0.81 APLNR (0.58) APLNRTAS2R14L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3601297-B9 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN AMGEN INC (US) 2023-05-24 EP disclosed